General Information of the Compound
Compound ID
CP0569068
Compound Name
methyl (2S,4aR,6aR,7R,9S,10aS,10bR)-2-(furan-3-yl)-9-[4-(hydroxymethyl)benzoyl]oxy-6a,10b-dimethyl-4,10-dioxo-2,4a,5,6,7,8,9,10a-octahydro-1H-benzo[f]isochromene-7-carboxylate
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Structure
Formula
C29H32O9
Molecular Weight
524.566
Canonical SMILES
COC(=O)[C@@H]1C[C@H](OC(=O)c2ccc(CO)cc2)C(=O)[C@H]2[C@@]1(C)CC[C@H]1C(=O)O[C@@H](C[C@]21C)c1ccoc1
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InChI
InChI=1S/C29H32O9/c1-28-10-8-19-27(34)38-22(18-9-11-36-15-18)13-29(19,2)24(28)23(31)21(12-20(28)26(33)35-3)37-25(32)17-6-4-16(14-30)5-7-17/h4-7,9,11,15,19-22,24,30H,8,10,12-14H2,1-3H3/t19-,20-,21-,22-,24-,28-,29-/m0/s1
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InChIKey
GAFSLIGIDICZRF-UTFYOTOKSA-N
Physicochemical Property
logP
3.7863
Rotatable Bonds
5
Heavy Atom Count
38
Polar Areas
129.34
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
9
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168282272
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 0.03 nM
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