General Information of the Compound
Compound ID
CP0555516
Compound Name
N-[4-[1-[2-[2-[2-[2-[2-[2-[4-[4-[2,3-dihydro-1H-inden-2-yl(propyl)amino]butyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]butyl]-N-propyl-2,3-dihydro-1H-inden-2-amine
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Formula
C48H74N8O5
Molecular Weight
843.171
Canonical SMILES
CCCN(CCCCc1cn(CCOCCOCCOCCOCCOCCn2cc(CCCCN(CCC)C3Cc4ccccc4C3)nn2)nn1)C1Cc2ccccc2C1
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InChI
InChI=1S/C48H74N8O5/c1-3-19-53(47-35-41-13-5-6-14-42(41)36-47)21-11-9-17-45-39-55(51-49-45)23-25-57-27-29-59-31-33-61-34-32-60-30-28-58-26-24-56-40-46(50-52-56)18-10-12-22-54(20-4-2)48-37-43-15-7-8-16-44(43)38-48/h5-8,13-16,39-40,47-48H,3-4,9-12,17-38H2,1-2H3
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InChIKey
CGDGQEFCZTTZBO-UHFFFAOYSA-N
Physicochemical Property
logP
6.057
Rotatable Bonds
34
Heavy Atom Count
61
Polar Areas
114.05
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
13
Complexity
61

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4755336
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 3.2 nM
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