General Information of the Compound
Compound ID
CP0551344
Compound Name
US8969325, 153
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Structure
Formula
C21H20F4N4O3
Molecular Weight
452.408
Canonical SMILES
CN1C(=O)NCc2c(NC(=O)N[C@@H]3CC(CF)(CF)Oc4c(F)cc(F)cc34)cccc12
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InChI
InChI=1S/C21H20F4N4O3/c1-29-17-4-2-3-15(13(17)8-26-20(29)31)27-19(30)28-16-7-21(9-22,10-23)32-18-12(16)5-11(24)6-14(18)25/h2-6,16H,7-10H2,1H3,(H,26,31)(H2,27,28,30)/t16-/m1/s1
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InChIKey
UHZPZFHAXSAGIS-MRXNPFEDSA-N
Physicochemical Property
logP
3.9473
Rotatable Bonds
4
Heavy Atom Count
32
Polar Areas
82.7
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
3
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 89647022
ChEMBL ID
CHEMBL3682242
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02183, Transient receptor potential cation channel subfamily V member 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 170 nM
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