General Information of the Compound
Compound ID
CP0549145
Compound Name
5-[5-[2-(1-methylpiperidin-4-yl)oxypyrimidin-5-yl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile
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Structure
Formula
C23H22F3N7O2S
Molecular Weight
517.537
Canonical SMILES
CN1CCC(CC1)Oc1ncc(cn1)N1C(=S)N(C(=O)C11CCC1)c1cnc(C#N)c(c1)C(F)(F)F
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InChI
InChI=1S/C23H22F3N7O2S/c1-31-7-3-16(4-8-31)35-20-29-12-15(13-30-20)33-21(36)32(19(34)22(33)5-2-6-22)14-9-17(23(24,25)26)18(10-27)28-11-14/h9,11-13,16H,2-8H2,1H3
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InChIKey
FETCXMHYNSCFGK-UHFFFAOYSA-N
Physicochemical Property
logP
3.29588
Rotatable Bonds
4
Heavy Atom Count
36
Polar Areas
98.48
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
8
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 130229412
ChEMBL ID
CHEMBL4850003
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00894, Androgen receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000141 LNCaP Homo sapiens (Human)  2
1
IC50 = 417 nM
   TI
   LI
   LO
   TS
2
IC50 = 427 nM
   TI
   LI
   LO
   TS