General Information of the Compound
Compound ID
CP0523759
Compound Name
1-[(R)-1-(2,4-Dichloro-benzyl)-2-oxo-2-(4-{2-[(2-thiophen-2-yl-ethylamino)-methyl]-phenyl}-piperazin-1-yl)-ethyl]-3-(2-fluoro-benzyl)-urea
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Structure
Formula
C34H36Cl2FN5O2S
Molecular Weight
668.666
Canonical SMILES
Fc1ccccc1CNC(=O)N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1CCN(CC1)c1ccccc1CNCCc1cccs1
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InChI
InChI=1S/C34H36Cl2FN5O2S/c35-27-12-11-24(29(36)21-27)20-31(40-34(44)39-23-25-6-1-3-9-30(25)37)33(43)42-17-15-41(16-18-42)32-10-4-2-7-26(32)22-38-14-13-28-8-5-19-45-28/h1-12,19,21,31,38H,13-18,20,22-23H2,(H2,39,40,44)/t31-/m1/s1
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InChIKey
CJYACAQSCXVWGG-WJOKGBTCSA-N
Physicochemical Property
logP
6.2856
Rotatable Bonds
12
Heavy Atom Count
45
Polar Areas
76.71
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
5
Complexity
45

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44400812
ChEMBL ID
CHEMBL195734
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00914, Melanocortin receptor 4
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 5 nM
   TI
   LI
   LO
   TS
Protein ID: PT01804, Melanocortin receptor 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 2300 nM
   TI
   LI
   LO
   TS