General Information of the Compound
Compound ID
CP0521706
Compound Name
(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[2-[[(2S,3S)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-2-[[2-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]acetyl]amino]propanoyl]amino]acetyl]amino]butanediamide
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Structure
Formula
C65H109N21O17
Molecular Weight
1456.717
Canonical SMILES
CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@H](C)NC(=O)CNC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(N)=O
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InChI
InChI=1S/C65H109N21O17/c1-15-34(10)52(64(102)84-44(19-33(8)9)63(101)86-53(38(14)87)65(103)80-42(54(68)92)17-31(4)5)85-51(91)27-72-56(94)36(12)77-57(95)37(13)78-60(98)46(21-40-24-70-29-75-40)83-62(100)47(22-48(67)88)79-50(90)26-71-55(93)35(11)76-49(89)25-73-59(97)45(20-39-23-69-28-74-39)82-61(99)43(18-32(6)7)81-58(96)41(66)16-30(2)3/h23-24,28-38,41-47,52-53,87H,15-22,25-27,66H2,1-14H3,(H2,67,88)(H2,68,92)(H,69,74)(H,70,75)(H,71,93)(H,72,94)(H,73,97)(H,76,89)(H,77,95)(H,78,98)(H,79,90)(H,80,103)(H,81,96)(H,82,99)(H,83,100)(H,84,102)(H,85,91)(H,86,101)/t34-,35-,36-,37-,38+,41-,42-,43-,44-,45-,46-,47-,52-,53-/m0/s1
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InChIKey
NNVHPEYZHVLEFM-ZWGHFTKOSA-N
Physicochemical Property
logP
-6.0416
Rotatable Bonds
46
Heavy Atom Count
103
Polar Areas
597.19
Hydrogen Bond Donor Count
20
Hydrogen Bond Acceptor Count
20
Complexity
103

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44376981
ChEMBL ID
CHEMBL265424
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000076 CHO/Galpha16 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 947 nM
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Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000076 CHO/Galpha16 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 1380 nM
   TI
   LI
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   TS