General Information of the Compound
Compound ID
CP0491435
Compound Name
5-[8-oxo-5-(2-piperidin-4-yloxypyrimidin-5-yl)-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile
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Structure
Formula
C22H20F3N7O2S
Molecular Weight
503.51
Canonical SMILES
FC(F)(F)c1cc(cnc1C#N)N1C(=S)N(c2cnc(OC3CCNCC3)nc2)C2(CCC2)C1=O
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InChI
InChI=1S/C22H20F3N7O2S/c23-22(24,25)16-8-13(10-28-17(16)9-26)31-18(33)21(4-1-5-21)32(20(31)35)14-11-29-19(30-12-14)34-15-2-6-27-7-3-15/h8,10-12,15,27H,1-7H2
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InChIKey
QWTUBLVEMRHUOG-UHFFFAOYSA-N
Physicochemical Property
logP
2.95368
Rotatable Bonds
4
Heavy Atom Count
35
Polar Areas
107.27
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 130228990
ChEMBL ID
CHEMBL4868340
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00894, Androgen receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000141 LNCaP Homo sapiens (Human)  2
1
IC50 = 309 nM
   TI
   LI
   LO
   TS
2
IC50 = 501 nM
   TI
   LI
   LO
   TS