General Information of the Compound
Compound ID
CP0478048
Compound Name
CHEMBL4129031
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Formula
C24H25NO6
Molecular Weight
423.465
Canonical SMILES
CCOC(=O)c1ccc(cc1)N1C(C(C)C)C(C(=O)c2ccc(OC)cc2)=C(O)C1=O
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InChI
InChI=1S/C24H25NO6/c1-5-31-24(29)16-6-10-17(11-7-16)25-20(14(2)3)19(22(27)23(25)28)21(26)15-8-12-18(30-4)13-9-15/h6-14,20,27H,5H2,1-4H3
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InChIKey
IYCZOMGTSUJAMH-UHFFFAOYSA-N
Physicochemical Property
logP
3.9381
Rotatable Bonds
7
Heavy Atom Count
31
Polar Areas
93.14
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
SID: 56417081
ChEMBL ID
CHEMBL4129031
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03393, P2X purinoceptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000093 C6-BU-1 Rattus norvegicus (Rat)  1
1
IC50 = 140 nM
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