General Information of the Compound
Compound ID
CP0449809
Compound Name
(3-chloro-4-fluorophenyl)-[4-fluoro-4-[[[6-(1H-pyrazol-5-yl)pyridin-2-yl]methylamino]methyl]piperidin-1-yl]methanone
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Structure
Formula
C22H22ClF2N5O
Molecular Weight
445.901
Canonical SMILES
Fc1ccc(cc1Cl)C(=O)N1CCC(F)(CNCc2cccc(n2)-c2cc[nH]n2)CC1
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InChI
InChI=1S/C22H22ClF2N5O/c23-17-12-15(4-5-18(17)24)21(31)30-10-7-22(25,8-11-30)14-26-13-16-2-1-3-19(28-16)20-6-9-27-29-20/h1-6,9,12,26H,7-8,10-11,13-14H2,(H,27,29)
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InChIKey
MPFWDYYEEJVUMZ-UHFFFAOYSA-N
Physicochemical Property
logP
3.9983
Rotatable Bonds
6
Heavy Atom Count
31
Polar Areas
73.91
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
4
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10694660
SID: 15728646
ChEMBL ID
CHEMBL46539
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00819, 5-hydroxytryptamine receptor 1A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000803 HA7 Homo sapiens (Human)  1
1
EC50 = 0.7244 nM
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