General Information of the Compound
Compound ID
CP0438786
Compound Name
N-[4-[2-(3,3-difluoropyrrolidin-1-yl)ethoxy]-3-(2-methylpyrazol-3-yl)phenyl]-3-(trifluoromethyl)benzamide
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Structure
Formula
C24H23F5N4O2
Molecular Weight
494.464
Canonical SMILES
Cn1nccc1-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1OCCN1CCC(F)(F)C1
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InChI
InChI=1S/C24H23F5N4O2/c1-32-20(7-9-30-32)19-14-18(31-22(34)16-3-2-4-17(13-16)24(27,28)29)5-6-21(19)35-12-11-33-10-8-23(25,26)15-33/h2-7,9,13-14H,8,10-12,15H2,1H3,(H,31,34)
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InChIKey
UTGILOVPWVPYDC-UHFFFAOYSA-N
Physicochemical Property
logP
5.078
Rotatable Bonds
7
Heavy Atom Count
35
Polar Areas
59.39
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 46833072
SID: 99210961
ChEMBL ID
CHEMBL1083449
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00825, 5-hydroxytryptamine receptor 2A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 12 nM
   TI
   LI
   LO
   TS
Protein ID: PT00939, 5-hydroxytryptamine receptor 2C
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 9250 nM
   TI
   LI
   LO
   TS