General Information of the Compound
Compound ID
CP0432400
Compound Name
[(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[7-(hydroxyamino)-7-oxoheptanoyl]piperazine-1-carboxylate
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Structure
Formula
C34H39N5O9
Molecular Weight
661.712
Canonical SMILES
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCC(=O)NO)cc12
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InChI
InChI=1S/C34H39N5O9/c1-3-21-22-16-20(48-33(44)38-14-12-37(13-15-38)29(41)9-7-5-6-8-28(40)36-46)10-11-26(22)35-30-23(21)18-39-27(30)17-25-24(31(39)42)19-47-32(43)34(25,45)4-2/h10-11,16-17,45-46H,3-9,12-15,18-19H2,1-2H3,(H,36,40)/t34-/m0/s1
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InChIKey
YNXNNJTYDYSDAY-UMSFTDKQSA-N
Physicochemical Property
logP
2.7409
Rotatable Bonds
9
Heavy Atom Count
48
Polar Areas
180.6
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
11
Complexity
48

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145982778
ChEMBL ID
CHEMBL4241995
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00991, Histone deacetylase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 13620 nM
   TI
   LI
   LO
   TS
Protein ID: PT00995, Histone deacetylase 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS