General Information of the Compound
Compound ID
CP0415234
Compound Name
US8853203, 61
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Structure
Formula
C20H22N4O2
Molecular Weight
350.422
Canonical SMILES
COc1cccc2C3=CC(=NCC(=O)N3CCc12)n1cnc(c1)C(C)C
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InChI
InChI=1S/C20H22N4O2/c1-13(2)16-11-23(12-22-16)19-9-17-14-5-4-6-18(26-3)15(14)7-8-24(17)20(25)10-21-19/h4-6,9,11-13H,7-8,10H2,1-3H3
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InChIKey
KYTHQUHMVMDEQH-UHFFFAOYSA-N
Physicochemical Property
logP
2.7011
Rotatable Bonds
2
Heavy Atom Count
26
Polar Areas
59.72
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
5
Complexity
26

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 73335545
ChEMBL ID
CHEMBL3702409
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01994, Metabotropic glutamate receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000101 L-M(TK-) Mus musculus (Mouse)  1
1
IC50 = 3100 nM
   TI
   LI
   LO
   TS
Protein ID: PT00854, Metabotropic glutamate receptor 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000101 L-M(TK-) Mus musculus (Mouse)  1
1
IC50 = 345 nM
   TI
   LI
   LO
   TS