General Information of the Compound
Compound ID
CP0404107
Compound Name
(5S,8R,11S,14S,17S)-8-benzyl-11-[3-(diaminomethylideneamino)propyl]-5-(1H-imidazol-5-ylmethyl)-14-(1H-indol-3-ylmethyl)-2,2-dimethyl-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadecane-17-carboxamide
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Structure
Formula
C40H51N13O7
Molecular Weight
825.932
Canonical SMILES
CC1(C)NC(=O)C[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC1=O)C(N)=O
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InChI
InChI=1S/C40H51N13O7/c1-40(2)38(60)52-31(17-24-20-44-21-47-24)37(59)50-29(15-22-9-4-3-5-10-22)35(57)48-27(13-8-14-45-39(42)43)34(56)51-30(16-23-19-46-26-12-7-6-11-25(23)26)36(58)49-28(33(41)55)18-32(54)53-40/h3-7,9-12,19-21,27-31,46H,8,13-18H2,1-2H3,(H2,41,55)(H,44,47)(H,48,57)(H,49,58)(H,50,59)(H,51,56)(H,52,60)(H,53,54)(H4,42,43,45)/t27-,28-,29+,30-,31-/m0/s1
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InChIKey
CJCOTNMGGCNQIS-YSLHKSLUSA-N
Physicochemical Property
logP
-1.61003
Rotatable Bonds
11
Heavy Atom Count
60
Polar Areas
324.06
Hydrogen Bond Donor Count
12
Hydrogen Bond Acceptor Count
9
Complexity
60

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145975465
ChEMBL ID
CHEMBL4207725
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01325, Melanocortin receptor 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 76 nM
   TI
   LI
   LO
   TS
2
IC50 = 20 nM
   TI
   LI
   LO
   TS
Protein ID: PT00914, Melanocortin receptor 4
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 6.7 nM
   TI
   LI
   LO
   TS
2
IC50 = 5.2 nM
   TI
   LI
   LO
   TS
Protein ID: PT01804, Melanocortin receptor 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 140 nM
   TI
   LI
   LO
   TS
2
IC50 > 1000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00911, Melanocyte-stimulating hormone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 87 nM
   TI
   LI
   LO
   TS
2
IC50 = 601 nM
   TI
   LI
   LO
   TS