General Information of the Compound
Compound ID
CP0392297
Compound Name
tert-butyl (3S)-3-[(8-chloro-11-ethyl-3-fluoro-5H-benzo[b][1,4]benzodiazepin-6-ylidene)amino]pyrrolidine-1-carboxylate
    Show/Hide
Structure
Formula
C24H28ClFN4O2
Molecular Weight
458.965
Canonical SMILES
CCN1c2ccc(F)cc2N=C(N[C@H]2CCN(C2)C(=O)OC(C)(C)C)c2cc(Cl)ccc12
    Show/Hide
InChI
InChI=1S/C24H28ClFN4O2/c1-5-30-20-8-6-15(25)12-18(20)22(28-19-13-16(26)7-9-21(19)30)27-17-10-11-29(14-17)23(31)32-24(2,3)4/h6-9,12-13,17H,5,10-11,14H2,1-4H3,(H,27,28)/t17-/m0/s1
    Show/Hide
InChIKey
GKEGWJJRPYLMOW-KRWDZBQOSA-N
Physicochemical Property
logP
5.6278
Rotatable Bonds
2
Heavy Atom Count
32
Polar Areas
57.17
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 137125257
ChEMBL ID
CHEMBL3609370
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01042, Serine/threonine-protein kinase PAK 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd = 130 nM
   TI
   LI
   LO
   TS
Protein ID: PT01573, Serine/threonine-protein kinase PAK 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd > 40000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01076, Serine/threonine-protein kinase PAK 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd > 40000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01317, Serine/threonine-protein kinase PAK 4
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd > 40000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01413, Serine/threonine-protein kinase PAK 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd > 40000 nM
   TI
   LI
   LO
   TS