General Information of the Compound
Compound ID
CP0382523
Compound Name
2-(3-(methylamino)pyrrolidin-1-yl)-N-(4-(trifluoromethyl)phenyl)-7-(3-(trifluoromethyl)pyridin-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[5,4-d]azepin-4-amine
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Structure
Formula
C26H27F6N7
Molecular Weight
551.539
Canonical SMILES
CNC1CCN(C1)c1nc2CCN(CCc2c(Nc2ccc(cc2)C(F)(F)F)n1)c1ncccc1C(F)(F)F
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InChI
InChI=1S/C26H27F6N7/c1-33-18-8-12-39(15-18)24-36-21-10-14-38(23-20(26(30,31)32)3-2-11-34-23)13-9-19(21)22(37-24)35-17-6-4-16(5-7-17)25(27,28)29/h2-7,11,18,33H,8-10,12-15H2,1H3,(H,35,36,37)
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InChIKey
VXNXKOQHRMWNCX-UHFFFAOYSA-N
Physicochemical Property
logP
5.0561
Rotatable Bonds
5
Heavy Atom Count
39
Polar Areas
69.21
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 53325956
ChEMBL ID
CHEMBL1629722
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02183, Transient receptor potential cation channel subfamily V member 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2790 nM
   TI
   LI
   LO
   TS
Protein ID: PT01914, Transient receptor potential cation channel subfamily V member 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS