General Information of the Compound
Compound ID
CP0226933
Compound Name
US11059828, Example 382
    Show/Hide
Synonyms
((3aR,6aS)-5-(4,6-dimethylpyrimidin- 2-yl)hexahydropyrrolo(3,4-c)pyrrol-2(1H)-yl)(2
1293281-49-8
AKOS032954213
BDBM118454
CHEMBL3597971
GTPL9308
JNJ-922
MIN-202
Methanone, (5-(4,6-dimethyl-2-pyrimidinyl)hexahydropyrrolo(3,4-C)pyrrol-2(1H)-yl)(2-fluoro-6-(2H-1,2,3-triazol-2-yl)phenyl)-
SCHEMBL1671257
SQOCEMCKYDVLMM-UHFFFAOYSA-N
Seltorexant
Seltorexant [USAN]
US8653263, 107
[2-(4,6-dimethylpyrimidin-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[2-fluoro-6-(triazol-2-yl)phenyl]methanone
    Show/Hide
Structure
Formula
C21H22FN7O
Molecular Weight
407.453
Canonical SMILES
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
    Show/Hide
InChI
InChI=1S/C21H22FN7O/c1-13-8-14(2)26-21(25-13)28-11-15-9-27(10-16(15)12-28)20(30)19-17(22)4-3-5-18(19)29-23-6-7-24-29/h3-8,15-16H,9-12H2,1-2H3
    Show/Hide
InChIKey
SQOCEMCKYDVLMM-UHFFFAOYSA-N
CAS
1293281-49-8
Physicochemical Property
logP
2.02164
Rotatable Bonds
3
Heavy Atom Count
30
Polar Areas
80.04
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
7
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 67116280
ChEMBL ID
CHEMBL3597971
Clinical Information about the Compound
Drug 1 ( MIN-202 )
Drug Name MIN-202
Company Minerva Neurosciences Waltham, MA
Indication
Major depressive disorder
Phase 2
Target(s)
Orexin receptor type 2 (HCRTR2)
Antagonist