General Information of the Compound
Compound ID
CP0175608
Compound Name
N-[6-(3,4-dihydro-1H-isoquinolin-2-yl)-2-(3,5-dimethylpyrazol-1-yl)pyrimidin-4-yl]-1,3-thiazol-2-amine
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Structure
Formula
C21H21N7S
Molecular Weight
403.515
Canonical SMILES
Cc1cc(C)n(n1)-c1nc(Nc2nccs2)cc(n1)N1CCc2ccccc2C1
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InChI
InChI=1S/C21H21N7S/c1-14-11-15(2)28(26-14)20-23-18(24-21-22-8-10-29-21)12-19(25-20)27-9-7-16-5-3-4-6-17(16)13-27/h3-6,8,10-12H,7,9,13H2,1-2H3,(H,22,23,24,25)
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InChIKey
OQMYLASDAPUQRT-UHFFFAOYSA-N
Physicochemical Property
logP
4.04194
Rotatable Bonds
4
Heavy Atom Count
29
Polar Areas
71.76
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 72945317
ChEMBL ID
CHEMBL3100162
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 66 nM
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