General Information of the Compound
Compound ID
CP0172465
Compound Name
6-(3,4-dihydro-1H-isoquinolin-2-yl)-2-(3,5-dimethylpyrazol-1-yl)-N-pyrazin-2-ylpyrimidin-4-amine
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Structure
Formula
C22H22N8
Molecular Weight
398.474
Canonical SMILES
Cc1cc(C)n(n1)-c1nc(Nc2cnccn2)cc(n1)N1CCc2ccccc2C1
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InChI
InChI=1S/C22H22N8/c1-15-11-16(2)30(28-15)22-26-19(25-20-13-23-8-9-24-20)12-21(27-22)29-10-7-17-5-3-4-6-18(17)14-29/h3-6,8-9,11-13H,7,10,14H2,1-2H3,(H,24,25,26,27)
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InChIKey
CRGTXSAUQFYFSM-UHFFFAOYSA-N
Physicochemical Property
logP
3.37544
Rotatable Bonds
4
Heavy Atom Count
30
Polar Areas
84.65
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 72793900
ChEMBL ID
CHEMBL3100161
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1.1 nM
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