General Information of the Compound
Compound ID
CP0109572
Compound Name
3-[5-Chloro-4-(2-fluoro-6-methylcarbamoyl-phenylamino)-pyrimidin-2-ylamino]-7,8-dihydro-6H-5-oxa-9-aza-benzocycloheptene-9-carboxylic acid 2-methoxy-ethyl ester
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Structure
Formula
C25H26ClFN6O5
Molecular Weight
544.971
Canonical SMILES
CNC(=O)c1cccc(F)c1Nc1nc(Nc2ccc3N(CCCOc3c2)C(=O)OCCOC)ncc1Cl
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InChI
InChI=1S/C25H26ClFN6O5/c1-28-23(34)16-5-3-6-18(27)21(16)31-22-17(26)14-29-24(32-22)30-15-7-8-19-20(13-15)37-10-4-9-33(19)25(35)38-12-11-36-2/h3,5-8,13-14H,4,9-12H2,1-2H3,(H,28,34)(H2,29,30,31,32)
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InChIKey
DQILXXVPFRTBOV-UHFFFAOYSA-N
Physicochemical Property
logP
4.4878
Rotatable Bonds
8
Heavy Atom Count
38
Polar Areas
126.94
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
9
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 53321320
ChEMBL ID
CHEMBL1642139
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01201, Hepatocyte growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000282 GTL-16 Homo sapiens (Human)  1
1
IC50 = 50 nM
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