General Information of the Compound
Compound ID
CP0071673
Compound Name
N-[(3R)-8-[[5-chloro-4-[2-fluoro-6-(methylcarbamoyl)anilino]pyrimidin-2-yl]amino]-5,5-dimethyl-2-oxo-3,4-dihydro-1H-1-benzazepin-3-yl]pyrrolidine-1-carboxamide
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Synonyms
BDBM50361564
GTPL8213
PMID21967808CR-16
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Structure
Formula
C29H32ClFN8O3
Molecular Weight
595.079
Canonical SMILES
CNC(=O)c1cccc(F)c1Nc1nc(Nc2ccc3c(NC(=O)[C@@H](CC3(C)C)NC(=O)N3CCCC3)c2)ncc1Cl
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InChI
InChI=1S/C29H32ClFN8O3/c1-29(2)14-22(36-28(42)39-11-4-5-12-39)26(41)35-21-13-16(9-10-18(21)29)34-27-33-15-19(30)24(38-27)37-23-17(25(40)32-3)7-6-8-20(23)31/h6-10,13,15,22H,4-5,11-12,14H2,1-3H3,(H,32,40)(H,35,41)(H,36,42)(H2,33,34,37,38)/t22-/m1/s1
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InChIKey
HGSNUBHWAMMKIR-JOCHJYFZSA-N
Physicochemical Property
logP
4.9097
Rotatable Bonds
6
Heavy Atom Count
42
Polar Areas
140.38
Hydrogen Bond Donor Count
5
Hydrogen Bond Acceptor Count
7
Complexity
42

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 56597775
SID: 134331276
ChEMBL ID
CHEMBL1939491
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01201, Hepatocyte growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000282 GTL-16 Homo sapiens (Human)  1
1
IC50 = 26 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( PMID21967808CR-16 )
Drug Name PMID21967808CR-16
Target(s)
IL-1 receptor-associated kinase 3 (IRAK3)
Inhibitor
Sugen kinase 110 (SBK3)
Inhibitor
Serine/threonine-protein kinase ULK1 (ULK1)
Inhibitor
Proto-oncogene c-Met (MET)
Inhibitor
Tie-1 tyrosine kinase receptor (TIE1)
Inhibitor