General Information of the Compound
Compound ID
CP0060653
Compound Name
1-(4-(4-(3,6-dihydro-2H-pyran-4-yl)-1-(2,2,2-trifluoroethyl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)phenyl)-3-(2-fluoroethyl)urea
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Structure
Formula
C21H20F4N6O2
Molecular Weight
464.423
Canonical SMILES
FCCNC(=O)Nc1ccc(cc1)-c1nc(C2=CCOCC2)c2cnn(CC(F)(F)F)c2n1
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InChI
InChI=1S/C21H20F4N6O2/c22-7-8-26-20(32)28-15-3-1-14(2-4-15)18-29-17(13-5-9-33-10-6-13)16-11-27-31(19(16)30-18)12-21(23,24)25/h1-5,11H,6-10,12H2,(H2,26,28,32)
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InChIKey
HAGVHIKZYFOZND-UHFFFAOYSA-N
Physicochemical Property
logP
3.9503
Rotatable Bonds
6
Heavy Atom Count
33
Polar Areas
93.96
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44156157
SID: 85156038
ChEMBL ID
CHEMBL590104
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01065, Serine/threonine-protein kinase mTOR
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1 nM
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