General Information of the Compound
Compound ID
CP0025347
Compound Name
(S)-2-(3-(3-hydroxy-5-methylphenyl)-4-(6-(2-hydroxypropylamino)-2-(pyridin-3-yl)pyrimidin-4-yl)-1H-pyrazol-1-yl)acetonitrile
    Show/Hide
Structure
Formula
C24H23N7O2
Molecular Weight
441.495
Canonical SMILES
C[C@H](O)CNc1cc(nc(n1)-c1cccnc1)-c1cn(CC#N)nc1-c1cc(C)cc(O)c1
    Show/Hide
InChI
InChI=1S/C24H23N7O2/c1-15-8-18(10-19(33)9-15)23-20(14-31(30-23)7-5-25)21-11-22(27-12-16(2)32)29-24(28-21)17-4-3-6-26-13-17/h3-4,6,8-11,13-14,16,32-33H,7,12H2,1-2H3,(H,27,28,29)/t16-/m0/s1
    Show/Hide
InChIKey
XNRABRXYGRUDAX-INIZCTEOSA-N
Physicochemical Property
logP
3.3994
Rotatable Bonds
7
Heavy Atom Count
33
Polar Areas
132.77
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
9
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 44517769
SID: 85853001
ChEMBL ID
CHEMBL560733
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01061, Proto-oncogene tyrosine-protein kinase ROS
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000310 HCC78 Homo sapiens (Human)  1
1
IC50 = 775 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 1.7 nM
2 IC50 = 199 nM