General Information of the Compound
Compound ID
CP0014446
Compound Name
N-[2-[2-[2-[2-[4-[[2-methoxy-4-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]phenoxy]methyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethyl]-2-[5-[2-(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridin-3-yl]oxyacetamide
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Structure
Formula
C43H52N8O8S
Molecular Weight
841.004
Canonical SMILES
COc1ccccc1N1CCN(Cc2ccc(OCc3cn(CCOCCOCCOCCNC(=O)COc4cncc(c4)C#Cc4csc(C)n4)nn3)c(OC)c2)CC1
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InChI
InChI=1S/C43H52N8O8S/c1-33-46-36(32-60-33)10-8-34-24-38(27-44-26-34)58-31-43(52)45-12-18-55-20-22-57-23-21-56-19-17-51-29-37(47-48-51)30-59-41-11-9-35(25-42(41)54-3)28-49-13-15-50(16-14-49)39-6-4-5-7-40(39)53-2/h4-7,9,11,24-27,29,32H,12-23,28,30-31H2,1-3H3,(H,45,52)
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InChIKey
SIMRHOCKDXANLH-UHFFFAOYSA-N
Physicochemical Property
logP
4.00122
Rotatable Bonds
23
Heavy Atom Count
60
Polar Areas
156.68
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
16
Complexity
60

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145984337
ChEMBL ID
CHEMBL4249547
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  2
1
Ki = 251 nM
   TI
   LI
   LO
   TS
2
Ki = 438 nM
   TI
   LI
   LO
   TS
Protein ID: PT00854, Metabotropic glutamate receptor 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 1200 nM
   TI
   LI
   LO
   TS