| Compound ID |
Compound Name |
Compound Formula |
|
CP0253387
|
(2S)-1-{(2S)-3-(1-methyl-1H-4-imidazolyl)-2-[(2S)-6-oxohexahydro-2-pyridinylcarboxamido]propanoyl}azolane-2-carboxamide
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|
C18H26N6O4
|
1
|
| 1 |
EC50 = 2.4 nM
|
|
|
|
CP0253386
|
(2S)-1-{(2S)-3-(1-ethyl-1H-4-imidazolyl)-2-[(2S)-6-oxohexahydro-2-pyridinylcarboxamido]propanoyl}azoazolane-2-carboxamide
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|
C19H28N6O4
|
1
|
| 1 |
EC50 = 2.8 nM
|
|
|
|
CP0067202
|
1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyrrolylcarboxamido)propanoyl]tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C16H22N6O4
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0408102
|
1-[2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-3-(2-propyl-1H-4-imidazolyl)-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C19H28N6O4
|
2
|
| 1 |
EC50 = 24 nM
|
|
|
| 2 |
Ki = 17000 nM
|
|
|
|
CP0162470
|
(2S)-1-[(2S)-2-(2S)-6-oxohexahydro-2-pyridinylcarboxamido]-3-(2-propyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C20H30N6O4
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0162668
|
(2S)-1-{(2S)-3-(1-allyl-1H-4-imidazolyl)-2-[(2S)-6-oxohexahydro-2-pyridinylcarboxamido]propropanoyl}azolane-2-carboxamide
Show/Hide
|
C20H28N6O4
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0497471
|
1-[3-(2-cyclopropyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C19H26N6O4
|
2
|
| 1 |
EC50 = 410 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0393980
|
1-[3-(2-cyclohexyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C22H32N6O4
|
2
|
| 1 |
EC50 = 1100 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0381542
|
1-[3-[2-(tert-butyl)-1H-4-imidazolyl]-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C20H30N6O4
|
2
|
| 1 |
EC50 = 1300 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0431207
|
1-[3-(2-isopropyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C19H28N6O4
|
2
|
| 1 |
EC50 = 1500 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0359955
|
(2S)-1-[(2S)-2-(2S)-6-oxohexahydro-2-pyridinylcarboxamido]-3-(2-isopropyl-1H-imidazolyl)propanoyl]-azalone-2-carboxamide
Show/Hide
|
C20H30N6O4
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
|
CP0359956
|
(2S)-1-{(2S)-3-(1-benzyl-1H-4-imidazolyl)-2-[(2S)-6-oxohexahydro-2-pyridinylcarboxamido]azolane-propanoyl}azolane-2-carboxamide
Show/Hide
|
C24H30N6O4
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0162460
|
(2S)-1-[(2S)-2-(2S)-6-oxohexahydro-2-pyridinylcarboxamido]-3-(2-tert-butyl-1H-imidazolyl)propanoyl]-azalone-2-carboxamide
Show/Hide
|
C21H32N6O4
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
|
CP0391620
|
1-[3-{2-[1-(1-adamantyl)ethyl]-1H-4-imidazolyl}-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
Show/Hide
|
C26H36N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0157755
|
(2S)-1-[(2S)-2-(1S)-3-oxocyclopentylcarboxamido]-3-(2-tert-butyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C21H31N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0157756
|
(2S)-1-[(2S)-2-(1R)-3-oxocyclopentylcarboxamido]-3-(2-propyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C20H29N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0162459
|
(2S)-1-[(2S)-2-(2S)-6-oxohexahydro-2-pyridinylcarboxamido]-3-(2-cyclohexyl-1H-imidazolyl)propanoyl]-azalone-2-carboxamide
Show/Hide
|
C23H34N6O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0253385
|
(2S)-1-[(2S)-2-(1R)-3-oxocyclopentylcarboxamido]-3-(2-tert-butyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C21H31N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0253388
|
(2S)-1-[(2S)-2-(1S)-3-oxocyclopentylcarboxamido]-3-(2-propyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C20H29N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0307083
|
(2S)-1-[(2S)-2-(1S)-3-oxocyclopentylcarboxamido]-3-(2-isopropyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C20H29N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0335691
|
(2S)-1-[(2S)-2-(1S)-3-oxocyclopentylcarboxamido]-3-(2-cyclohexyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C23H33N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0335692
|
(2S)-1-[(2S)-2-(1R)-3-oxocyclopentylcarboxamido]-3-(2-cyclohexyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C23H33N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0339773
|
(2S)-1-[(2S)-2-(1R)-3-oxocyclopentylcarboxamido]-3-(2-isopropyl-1H-imidazolyl)propanoyl]azalone-2-carboxamide
Show/Hide
|
C20H29N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
