Compound ID |
Compound Name |
Compound Formula |
CP0088908
|
N-benzyl-3-ethyl-6-[(2-methoxyacetyl)amino]-2-pyridin-3-ylbenzimidazole-4-carboxamide
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|
C25H25N5O3
|
1
|
1 |
IC50 = 3670 nM
|
|
|
CP0415169
|
1-[(2S)-2-hydroxy-3-[4-methoxy-2-[(2-pyridin-3-ylethylamino)methyl]phenoxy]propyl]piperidin-4-ol
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|
C23H33N3O4
|
1
|
1 |
IC50 = 4180 nM
|
|
|
CP0968706
|
(R)-4-(4-(3-hydroxy-3-methylbut-1-ynyl)benzyl)-1-((1-methyl-1H-pyrazol-4-yl)methyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
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|
C28H33N5O3
|
1
|
1 |
IC50 = 4250 nM
|
|
|
CP0559936
|
3-[(3S)-1-[[5-(3-hydroxy-3-methylbut-1-ynyl)thiophen-2-yl]methyl]piperidin-3-yl]-1-morpholin-4-ylpropan-1-one
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|
C22H32N2O3S
|
1
|
1 |
IC50 = 4420 nM
|
|
|
CP0376107
|
(5S)-5-[3-[4-[(R)-hydroxy(pyridin-3-yl)methyl]piperidin-1-yl]-3-oxopropyl]-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
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|
C29H33N3O3
|
1
|
1 |
IC50 = 23640 nM
|
|
|
CP0180984
|
2-[5-[bis(3-keto-5-methyl-3-pyrazolin-4-yl)methyl]-2-furyl]benzoic acid
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|
C20H18N4O5
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0482682
|
(3R)-N-[(3-fluorophenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
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|
C20H26FN3O3
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0866893
|
(S)-2-((R)-2-benzamido-3-(benzo[d][1,3]dioxol-5-yl)propanamido)-3-(1H-indol-3-yl)propanoic acid
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|
C28H25N3O6
|
1
|
1 |
IC50 = 100000 nM
|
|
|
CP0866894
|
(R)-6-(3-methoxybenzyloxy)-4-((S)-5-oxopyrrolidine-3-carbonyl)-1-phenethyl-1,4-diazepan-2-one
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|
C26H31N3O5
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0886161
|
(S)-2-(4-((5-methyl-1-propyl-1H-pyrazol-4-yl)methyl)-1-(3-phenylpropyl)piperazin-2-yl)ethanol
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|
C23H36N4O
|
1
|
1 |
IC50 > 100000 nM
|
|
|
CP0910693
|
N-benzyl-5-cyclopentyl-1-(2-hydroxyethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-3-carboxamide
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|
C21H28N4O2
|
1
|
1 |
IC50 > 100000 nM
|
|
|