| Compound ID |
Compound Name |
Compound Formula |
|
CP0514449
|
1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-one
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|
C22H29N3O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0460888
|
1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-azepan-2-one
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|
C23H31N3O2S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0447216
|
(S)-1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-pyrrolidine-2-carboxylic acid methyl ester
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|
C23H31N3O3S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0441282
|
1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-one; hydrochloride
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|
C24H33N3O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0418914
|
1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-pyrrolidin-2-one
Show/Hide
|
C21H27N3O2S
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0404209
|
1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-pyrrolidin-2-one
Show/Hide
|
C23H31N3O2S
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0436835
|
1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-1-methyl-1H-pyrazol-3-ylmethyl}-piperidin-2-one
Show/Hide
|
C24H35N5O2
|
1
|
| 1 |
Ki = 44 nM
|
|
|
|
CP0428734
|
1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-azepan-2-one
Show/Hide
|
C25H35N3O2S
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0451946
|
1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-2-methyl-2H-pyrazol-3-ylmethyl}-piperidin-2-one
Show/Hide
|
C24H35N5O2
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0424607
|
2-(2-oxopiperidin-1-yl)-N-[3-[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]propyl]acetamide
Show/Hide
|
C23H36N4O3
|
1
|
| 1 |
Ki = 80 nM
|
|
|
|
CP0401646
|
1-(5-Bromo-thiophen-2-ylmethyl)-4-(2-methoxy-phenyl)-piperazine
Show/Hide
|
C16H19BrN2OS
|
1
|
| 1 |
Ki = 92 nM
|
|
|
|
CP0479750
|
1-{5-[4-(2-Propoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-3-ylmethyl}-piperidin-2-one
Show/Hide
|
C24H33N3O2S
|
1
|
| 1 |
Ki = 92 nM
|
|
|
|
CP0441665
|
(2-Oxo-piperidin-1-yl)-acetic acid 2-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-ethyl ester
Show/Hide
|
C22H33N3O4
|
1
|
| 1 |
Ki = 108 nM
|
|
|
|
CP0437757
|
1-{5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophen-2-ylmethyl}-piperidin-2-ol
Show/Hide
|
C22H31N3O2S
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0441309
|
[5-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]thiophen-2-yl]methanol
Show/Hide
|
C17H22N2O2S
|
1
|
| 1 |
Ki = 138 nM
|
|
|
|
CP0415583
|
1-{5-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-2H-pyrazol-3-ylmethyl}-piperidin-2-one
Show/Hide
|
C23H33N5O2
|
1
|
| 1 |
Ki = 177 nM
|
|
|
|
CP0515889
|
1-{4-Hydroxy-5-[4-(2-isopropoxy-phenyl)-piperazin-1-yl]-2-oxo-pentyl}-piperidin-2-one
Show/Hide
|
C23H35N3O4
|
1
|
| 1 |
Ki = 253 nM
|
|
|
|
CP0501089
|
1-({2-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-ethylcarbamoyl}-methyl)-5-oxo-pyrrolidine-2-carboxylic acid ethyl ester
Show/Hide
|
C24H36N4O5
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0466836
|
5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-thiophene-2-carbaldehyde
Show/Hide
|
C17H20N2O2S
|
1
|
| 1 |
Ki = 262 nM
|
|
|
|
CP0380273
|
1-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-isoxazol-5-ylmethyl}-piperidin-2-one
Show/Hide
|
C23H32N4O3
|
1
|
| 1 |
Ki = 272 nM
|
|
|
|
CP0453097
|
[5-[[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]methyl]thiophen-3-yl]methanol
Show/Hide
|
C19H26N2O2S
|
1
|
| 1 |
Ki = 339 nM
|
|
|
|
CP0375998
|
2-(2-oxopiperidin-1-yl)-N-[2-[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]ethyl]acetamide
Show/Hide
|
C22H34N4O3
|
1
|
| 1 |
Ki = 372 nM
|
|
|
|
CP0497715
|
2-(2-oxoazepan-1-yl)-N-[2-[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]ethyl]acetamide
Show/Hide
|
C23H36N4O3
|
1
|
| 1 |
Ki = 505 nM
|
|
|
|
CP0921505
|
1-{(E)-5-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-2-oxo-pent-3-enyl}-piperidin-2-one
Show/Hide
|
C23H33N3O3
|
1
|
| 1 |
Ki = 602 nM
|
|
|
|
CP0497205
|
N-methyl-2-(2-oxopiperidin-1-yl)-N-[2-[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]ethyl]acetamide
Show/Hide
|
C23H36N4O3
|
1
|
| 1 |
Ki = 650 nM
|
|
|
|
CP0448732
|
1-{3-[4-(2-Isopropoxy-phenyl)-piperazin-1-ylmethyl]-4,5-dihydro-isoxazol-5-ylmethyl}-piperidin-2-one
Show/Hide
|
C23H34N4O3
|
1
|
| 1 |
Ki = 1517 nM
|
|
|
|
CP0419315
|
N-[2-[4-(4-fluoro-2-propan-2-yloxyphenyl)piperazin-1-yl]ethyl]-2-(2-oxopiperidin-1-yl)acetamide
Show/Hide
|
C22H33FN4O3
|
1
|
| 1 |
Ki = 4500 nM
|
|
|
|
CP0484760
|
N-[2-[4-[4-fluoro-2-(2,2,2-trifluoroethoxy)phenyl]piperazin-1-yl]ethyl]-2-(2-oxopiperidin-1-yl)acetamide
Show/Hide
|
C21H28F4N4O3
|
1
|
| 1 |
Ki = 5350 nM
|
|
|
|
CP0399342
|
1-[4-(2-Isopropoxy-phenyl)-piperazin-1-yl]-5-(2-oxo-piperidin-1-yl)-pentane-2,4-dione
Show/Hide
|
C23H33N3O4
|
1
|
| 1 |
Ki = 6043 nM
|
|
|
|
CP0374743
|
1-{2-Amino-6-[4-(2-isopropoxy-phenyl)-piperazin-1-ylmethyl]-pyrimidin-4-ylmethyl}-piperidin-2-one
Show/Hide
|
C24H34N6O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0505644
|
N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-2-(2-oxopiperidin-1-yl)acetamide
Show/Hide
|
C21H32N4O3
|
1
|
| 1 |
Ki = 10000 nM
|
|
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