Compound ID |
Compound Name |
Compound Formula |
CP0184261
|
N-cyclohexyl-2-(5-methyl-4-oxo-3,8-diphenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C31H30N4O2S
|
1
|
1 |
EC50 = 820 nM
|
|
|
CP0127752
|
N-cyclohexyl-2-(5-methyl-8-naphthalen-2-yl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C35H32N4O2S
|
1
|
1 |
EC50 = 2010 nM
|
|
|
CP0238282
|
2-(8-bromo-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanyl-N-cyclohexylacetamide
Show/Hide
|
C25H25BrN4O2S
|
1
|
1 |
EC50 = 2450 nM
|
|
|
CP0201870
|
N-cyclohexyl-2-(8-iodo-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C25H25IN4O2S
|
1
|
1 |
EC50 = 2510 nM
|
|
|
CP0184258
|
N-cyclohexyl-2-(5-methyl-8-naphthalen-1-yl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C35H32N4O2S
|
1
|
1 |
EC50 = 2580 nM
|
|
|
CP0476463
|
N-cyclohexyl-2-(8-ethynyl-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C27H26N4O2S
|
1
|
1 |
EC50 = 2740 nM
|
|
|
CP0303515
|
N-cyclohexyl-2-[(6-oxo-5-phenyl-3,5,8-triazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),3-trien-4-yl)sulfanyl]acetamide
Show/Hide
|
C25H30N4O2S
|
1
|
1 |
EC50 = 2830 nM
|
|
|
CP0127764
|
N-cyclohexyl-2-(5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanylacetamide
Show/Hide
|
C25H26N4O2S
|
1
|
1 |
EC50 = 3170 nM
|
|
|
CP0417558
|
N-cyclohexyl-2-[5-methyl-4-oxo-3-phenyl-8-(2-trimethylsilylethynyl)pyrimido[5,4-b]indol-2-yl]sulfanylacetamide
Show/Hide
|
C30H34N4O2SSi
|
1
|
1 |
EC50 = 3300 nM
|
|
|
CP0238283
|
2-(7-bromo-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanyl-N-cyclohexylacetamide
Show/Hide
|
C25H25BrN4O2S
|
1
|
1 |
EC50 = 4890 nM
|
|
|
CP0127750
|
N-cyclohexyl-2-[(4-oxo-3-phenyl-6,7,8,9-tetrahydro-5H-pyrimido[5,4-b]indol-2-yl)sulfanyl]acetamide
Show/Hide
|
C24H28N4O2S
|
1
|
1 |
EC50 = 7120 nM
|
|
|
CP0303517
|
N-cyclohexyl-2-[(8-methyl-6-oxo-5-phenyl-3,5,8-triazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),3-trien-4-yl)sulfanyl]acetamide
Show/Hide
|
C26H32N4O2S
|
1
|
1 |
EC50 = 8800 nM
|
|
|
CP0127749
|
N-cyclohexyl-2-[(5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)amino]acetamide
Show/Hide
|
C25H27N5O2
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0127751
|
N-cyclohexyl-2-[(6,7-dimethyl-4-oxo-3-phenyl-5H-pyrrolo[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H26N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0184256
|
N-[2-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-8-yl]benzamide
Show/Hide
|
C32H31N5O3S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0235985
|
2-(8-cyano-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanyl-N-cyclohexylacetamide
Show/Hide
|
C26H25N5O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0238280
|
N-cyclohexyl-2-[(5-methyl-4-oxo-3-phenyl-6,7,8,9-tetrahydropyrimido[5,4-b]indol-2-yl)sulfanyl]acetamide
Show/Hide
|
C25H30N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0238281
|
N-cyclohexyl-2-(5-methyl-4-oxo-3-phenylpyrrolo[3,2-d]pyrimidin-2-yl)sulfanylacetamide
Show/Hide
|
C21H24N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0303516
|
4-[[2-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-8-yl]amino]-4-oxobutanoic acid
Show/Hide
|
C29H31N5O5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0326610
|
2-(3-cyclohexylpropylsulfanyl)-3-phenyl-5H-pyrimido[5,4-b]indol-4-one
Show/Hide
|
C25H27N3OS
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0355546
|
2-(7-cyano-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanyl-N-cyclohexylacetamide
Show/Hide
|
C26H25N5O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0417555
|
N-cyclohexyl-2-[5-methyl-4-oxo-3-phenyl-8-(4-phenylphenyl)pyrimido[5,4-b]indol-2-yl]sulfanylacetamide
Show/Hide
|
C37H34N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0417570
|
N-[2-[2-(cyclohexylamino)-2-oxoethyl]sulfanyl-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-8-yl]octanamide
Show/Hide
|
C33H41N5O3S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0417571
|
N-cyclohexyl-2-(5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfonylacetamide
Show/Hide
|
C25H26N4O4S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0417572
|
N-cyclohexyl-2-(5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)oxyacetamide
Show/Hide
|
C25H26N4O3
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0448700
|
N-cyclohexyl-2-(5,6,7-trimethyl-4-oxo-3-phenylpyrrolo[3,2-d]pyrimidin-2-yl)sulfanylacetamide
Show/Hide
|
C23H28N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0448701
|
2-(8-amino-5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)sulfanyl-N-cyclohexylacetamide
Show/Hide
|
C25H27N5O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0448702
|
N-cyclohexyl-2-[(4-oxo-3-phenyl-5H-pyrrolo[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C20H22N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0475070
|
N-cyclohexyl-4-[(4-oxo-3-phenyl-5H-pyrimido[5,4-b]indol-2-yl)sulfanyl]butanamide
Show/Hide
|
C26H28N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0476464
|
N-cyclohexyl-3-[(5-methyl-4-oxo-3-phenylpyrimido[5,4-b]indol-2-yl)amino]propanamide
Show/Hide
|
C26H29N5O2
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0519697
|
N-cyclohexyl-3-[(4-oxo-3-phenyl-5H-pyrimido[5,4-b]indol-2-yl)sulfanyl]propanamide
Show/Hide
|
C25H26N4O2S
|
1
|
1 |
EC50 > 10000 nM
|
|
|