| Compound ID |
Compound Name |
Compound Formula |
|
CP0568137
|
[1-(cyclopropylmethyl)-4-(trifluoromethyl)pyrazolo[3,4-b]pyridin-5-yl]-[4-(2,4-difluorophenyl)piperazin-1-yl]methanone
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|
C22H20F5N5O
|
2
|
| 1 |
EC50 = 7.317 nM
|
|
|
| 2 |
EC50 = 84 nM
|
|
|
|
CP0568919
|
7-[[4-(4-chloro-2-fluorophenyl)piperazin-1-yl]methyl]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H22ClF4N5
|
2
|
| 1 |
EC50 = 8.3 nM
|
|
|
| 2 |
EC50 = 7278 nM
|
|
|
|
CP0544956
|
7-[[4-(2-chloro-4-fluorophenyl)piperazin-1-yl]methyl]-3-(cyclopropylmethyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H22ClF4N5
|
2
|
| 1 |
EC50 = 11 nM
|
|
|
| 2 |
EC50 = 2353 nM
|
|
|
|
CP0426536
|
(2S)-2-[[4-(2,3-dimethylphenyl)phenoxy]methyl]-6-ethyl-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C23H24N2O3
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0392578
|
(2S)-2-[[4-(2,3-dimethylphenyl)phenoxy]methyl]-6-methyl-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C22H22N2O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0458064
|
3-(cyclopropylmethyl)-7-[[4-(2,4-difluorophenyl)piperidin-1-yl]methyl]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C23H23F5N4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 371 nM
|
|
|
|
CP0046845
|
3-(cyclopropylmethyl)-7-[[4-(2,4-difluorophenyl)piperazin-1-yl]methyl]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H22F5N5
|
2
|
| 1 |
EC50 = 82 nM
|
|
|
| 2 |
EC50 = 166 nM
|
|
|
|
CP0544959
|
3-(cyclopropylmethyl)-8-[[4-(2,4-difluorophenyl)piperazin-1-yl]methyl]-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H22F5N5
|
2
|
| 1 |
EC50 = 136 nM
|
|
|
| 2 |
EC50 = 913 nM
|
|
|
|
CP0434655
|
(2S)-2-[(1,1-dimethyl-2,3-dihydroinden-5-yl)oxymethyl]-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C18H20N2O3
|
1
|
| 1 |
EC50 = 159 nM
|
|
|
|
CP0426559
|
(2S)-2-[[4-(2,3-dimethylphenyl)phenoxy]methyl]-5-methyl-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C22H22N2O3
|
1
|
| 1 |
EC50 = 274 nM
|
|
|
|
CP0392577
|
(2S)-2-[[4-(2,3-dimethylphenyl)phenoxy]methyl]-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C21H20N2O3
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0389392
|
(2S)-2-[(4-tert-butylphenoxy)methyl]-2,3-dihydro-[1,3]oxazolo[3,2-a]pyrimidin-7-one
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|
C17H20N2O3
|
1
|
| 1 |
EC50 = 1355 nM
|
|
|
|
CP0544958
|
3-(cyclopropylmethyl)-7-[[4-(2-fluorophenyl)piperazin-1-yl]methyl]-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H23F4N5
|
1
|
| 1 |
EC50 = 2089 nM
|
|
|
