| Compound ID |
Compound Name |
Compound Formula |
|
CP0530680
|
(11S)-5-ethyl-N-[(4-fluorophenyl)methyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
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|
C23H19FN2O3S
|
1
|
| 1 |
AC50 = 56 nM
|
|
|
|
CP0382130
|
(11S)-5-methyl-6,11-dioxo-N-(2-pyrrolidin-1-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
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|
C21H23N3O3S
|
1
|
| 1 |
AC50 = 70 nM
|
|
|
|
CP0382131
|
(11S)-5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
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|
C21H18N2O3S2
|
1
|
| 1 |
AC50 = 70 nM
|
|
|
|
CP0955852
|
rac-N-(4-Bromobenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C22H17BrN2O3S
|
1
|
| 1 |
AC50 = 71 nM
|
|
|
|
CP0411142
|
(11S)-N-[(4-bromophenyl)methyl]-5-methyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
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|
C22H17BrN2O3S
|
1
|
| 1 |
AC50 = 89 nM
|
|
|
|
CP0490048
|
5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
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|
C21H18N2O3S2
|
1
|
| 1 |
AC50 = 89 nM
|
|
|
|
CP0908021
|
rac-10-Methyl-11-oxo-N-(2-(pyrrolidin-1-yl)ethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C21H23N3O3S
|
1
|
| 1 |
AC50 = 89 nM
|
|
|
|
CP0913538
|
SID24383999
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|
C23H19FN2O3S
|
1
|
| 1 |
AC50 = 89 nM
|
|
|
|
CP0411141
|
(11S)-N-[(4-cyanophenyl)methyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
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|
C24H19N3O3S
|
1
|
| 1 |
AC50 = 112 nM
|
|
|
|
CP0864491
|
rac-N-(4-Methoxybenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C23H20N2O4S
|
1
|
| 1 |
AC50 = 112 nM
|
|
|
|
CP0951847
|
rac-10-Ethyl-N-(3-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C24H22N2O4S
|
1
|
| 1 |
AC50 = 112 nM
|
|
|
|
CP0955854
|
rac-10-Methyl-11-oxo-N-(2-(piperidin-1-yl)ethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C22H25N3O3S
|
1
|
| 1 |
AC50 = 112 nM
|
|
|
|
CP0864336
|
rac-10-Ethyl-11-oxo-N-(4-(trifluoromethyl)benzyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C24H19F3N2O3S
|
1
|
| 1 |
AC50 = 141 nM
|
|
|
|
CP0908023
|
10-Ethyl-N-(4-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-(S)-oxide
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|
C24H22N2O4S
|
1
|
| 1 |
AC50 = 141 nM
|
|
|
|
CP0913539
|
rac-N-(4-Cyanobenzyl)-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C24H19N3O3S
|
1
|
| 1 |
AC50 = 141 nM
|
|
|
|
CP0914735
|
rac-10-Ethyl-N-(4-methoxyphenyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C23H20N2O4S
|
1
|
| 1 |
AC50 = 141 nM
|
|
|
|
CP0939783
|
rac-N-(4-Chlorobenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C22H17ClN2O3S
|
1
|
| 1 |
AC50 = 141 nM
|
|
|
|
CP0793429
|
rac-10-Ethyl-N-(4-methylbenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C24H22N2O3S
|
1
|
| 1 |
AC50 = 177 nM
|
|
|
|
CP0480949
|
(11S)-N-[(1R)-1-(4-bromophenyl)ethyl]-5-ethyl-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
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|
C24H21BrN2O3S
|
1
|
| 1 |
AC50 = 223 nM
|
|
|
|
CP0864335
|
rac-N-(10-Ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepin-8-yl)-2-(4-fluorophenyl)acetamide 5-oxide
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|
C23H19FN2O3S
|
1
|
| 1 |
AC50 = 223 nM
|
|
|
|
CP0947327
|
rac-N-Benzyl-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H18N2O3S
|
1
|
| 1 |
AC50 = 223 nM
|
|
|
|
CP0956971
|
rac-10-Ethyl-N-(4-(methylthio)benzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C24H22N2O3S2
|
1
|
| 1 |
AC50 = 223 nM
|
|
|
|
CP0377527
|
5-ethyl-6,11-diketo-N-p-anisyl-benzo[b][1,4]benzothiazepine-3-carboxamide
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|
C24H22N2O4S
|
1
|
| 1 |
AC50 = 280 nM
|
|
|
|
CP0908024
|
N-(4-Chlorobenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-(S)-oxide
Show/Hide
|
C22H17ClN2O3S
|
1
|
| 1 |
AC50 = 280 nM
|
|
|
|
CP0914738
|
rac-N-(3-Chlorobenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H17ClN2O3S
|
1
|
| 1 |
AC50 = 281 nM
|
|
|
|
CP0957218
|
rac-10-Methyl-11-oxo-N-(pyridin-3-ylmethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C21H17N3O3S
|
1
|
| 1 |
AC50 = 281 nM
|
|
|
|
CP0380862
|
(11S)-5-ethyl-N-[(1R)-1-naphthalen-2-ylethyl]-6,11-dioxobenzo[b][1,4]benzothiazepine-3-carboxamide
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|
C28H24N2O3S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0848727
|
rac-N-(4-tert-Butylbenzyl)-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
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|
C27H28N2O3S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0848729
|
rac-N-(4-Fluorobenzyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H17FN2O3S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0849325
|
rac-10-Ethyl-N-(4-(methylsulfonyl)benzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C24H22N2O5S2
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0914736
|
rac-10-Ethyl-N-(4-methoxyphenethyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C25H24N2O4S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0914737
|
rac-N-(4-Methoxyphenyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H18N2O4S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0956973
|
rac-N-(benzo[d][1,3]dioxol-5-ylmethyl)-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C24H20N2O5S
|
1
|
| 1 |
AC50 = 353 nM
|
|
|
|
CP0411140
|
(11S)-5-methyl-6,11-dioxo-N-(pyridin-3-ylmethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
Show/Hide
|
C21H17N3O3S
|
1
|
| 1 |
AC50 = 445 nM
|
|
|
|
CP0953226
|
rac-N-Benzyl-10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C23H20N2O3S
|
1
|
| 1 |
AC50 = 445 nM
|
|
|
|
CP0908019
|
SID24383991
Show/Hide
|
C23H19ClN2O3S
|
1
|
| 1 |
AC50 = 509 nM
|
|
|
|
CP0848730
|
rac-N-(3-(Dimethylamino)propyl)-10-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C20H23N3O3S
|
1
|
| 1 |
AC50 = 560 nM
|
|
|
|
CP0914734
|
rac-10-Ethyl-11-oxo-N-(1-phenylethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C24H22N2O3S
|
1
|
| 1 |
AC50 = 560 nM
|
|
|
|
CP0848735
|
rac-N-(4-Methoxybenzyl)-11-oxo-10-propyl-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C25H24N2O4S
|
1
|
| 1 |
AC50 = 705 nM
|
|
|
|
CP0947328
|
rac-N-(10-Ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepin-8-yl)-2-(4-methoxyphenyl)acetamide 5-oxide
Show/Hide
|
C24H22N2O4S
|
1
|
| 1 |
AC50 = 705 nM
|
|
|
|
CP0956151
|
rac-10-Ethyl-N-(4-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide
Show/Hide
|
C24H22N2O3S
|
1
|
| 1 |
AC50 = 705 nM
|
|
|
|
CP0956596
|
rac-10-Ethyl-11-oxo-N-phenyl-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H18N2O3S
|
1
|
| 1 |
AC50 = 887 nM
|
|
|
|
CP0956597
|
rac-N-(4-Methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C22H18N2O4S
|
1
|
| 1 |
AC50 = 887 nM
|
|
|
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CP0848728
|
rac-10-Methyl-11-oxo-N-phenyl-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C21H16N2O3S
|
1
|
| 1 |
AC50 = 1580 nM
|
|
|
|
CP0956972
|
rac-10-Ethyl-11-oxo-N-(3,4,5-trimethoxybenzyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C26H26N2O6S
|
1
|
| 1 |
AC50 = 1770 nM
|
|
|
|
CP0956150
|
SID24383997
Show/Hide
|
C24H22N2O4S
|
1
|
| 1 |
AC50 = 4460 nM
|
|
|
|
CP0908020
|
SID24383931
Show/Hide
|
C29H24N2O4S
|
1
|
| 1 |
AC50 = 8870 nM
|
|
|
|
CP0955853
|
rac-10-Methyl-11-oxo-N-(pyridin-2-ylmethyl)-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C21H17N3O3S
|
1
|
| 1 |
AC50 = 11200 nM
|
|
|
|
CP0849327
|
rac-N-Benzyl-N,10-diethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C25H24N2O3S
|
1
|
| 1 |
AC50 = 56000 nM
|
|
|
|
CP0411143
|
(11R)-5-methyl-6,11-dioxo-N-(2-thiophen-2-ylethyl)benzo[b][1,4]benzothiazepine-3-carboxamide
Show/Hide
|
C21H18N2O3S2
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0848731
|
rac-4-Methoxybenzyl 10-ethyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxylate 5-oxide
Show/Hide
|
C24H21NO5S
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0849326
|
10-Ethyl-N-(4-methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-(R)-oxide
Show/Hide
|
C24H22N2O4S
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0908022
|
rac-10-Ethyl-N-(4-Methoxybenzyl)-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5,5-dioxide
Show/Hide
|
C24H22N2O5S
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0951855
|
rac-N-(4-Methoxybenzyl)-9,10-dioxo-9,10-dihydroanthracene-2-carboxamide
Show/Hide
|
C23H17NO4
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0951856
|
rac-10-Ethyl-N-(4-methoxybenzyl)-N-methyl-11-oxo-10,11-dihydrodibenzo[b,f][1,4]thiazepine-8-carboxamide 5-oxide
Show/Hide
|
C25H24N2O4S
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
|
CP0955855
|
rac-3-(1,3-Dioxoisoindolin-2-yl)-N-(4-methoxybenzyl)benzamide
Show/Hide
|
C23H18N2O4
|
1
|
| 1 |
AC50 > 77000 nM
|
|
|
