| Compound ID |
Compound Name |
Compound Formula |
|
CP0047806
|
6-chloro-2-oxo-N-((1R,3r,5S)-8-(((1-(4,4,4-trifluorobutyl)piperidin-4-yl)methyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)indoline-5-carboxamide
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|
C26H34ClF3N4O4S
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0047805
|
N-((1R,3r,5S)-8-((4-(benzylamino)piperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-6-chloro-2-oxoindoline-5-carboxamide
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|
C28H34ClN5O4S
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0566726
|
6-chloro-N-((1R,3r,5S)-8-((4-(dimethylamino)piperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C23H32ClN5O4S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0383126
|
N-((1R,3r,5S)-8-((4-aminopiperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-6-methyl-2-oxoindoline-5-carboxamide
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|
C22H31N5O4S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0447963
|
6-chloro-N-((1R,3r,5S)-8-((4-(methylamino)piperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C22H30ClN5O4S
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0414575
|
N-((1R,3r,5S)-8-(((1-methylpiperidin-4-yl)methyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C23H32N4O4S
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0566725
|
N-((1R,3r,5S)-8-((4-aminopiperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-6-fluoro-2-oxoindoline-5-carboxamide
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|
C21H28FN5O4S
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0414574
|
6-chloro-2-oxo-N-[(1S,5R)-8-[[(3R)-piperidin-3-yl]methylsulfonyl]-8-azabicyclo[3.2.1]octan-3-yl]-1,3-dihydroindole-5-carboxamide
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|
C22H29ClN4O4S
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0452624
|
6-chloro-N-((1R,3r,5S)-8-(((1-(3-hydroxypropyl)piperidin-4-yl)methyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C25H35ClN4O5S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0566724
|
N-((1R,3r,5S)-8-((4-aminopiperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C21H29N5O4S
|
1
|
| 1 |
IC50 = 850 nM
|
|
|
|
CP0472082
|
N-((1R,3r,5S)-8-((4-aminopiperidin-1-yl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-6-chloro-2-oxoindoline-5-carboxamide
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|
C21H28ClN5O4S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0475479
|
CHEMBL3798745
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|
C22H29ClN4O4S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0571195
|
N-((1R,3R,5S)-8-(((1r,4R)-4-aminocyclohexyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-2-oxoindoline-5-carboxamide
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|
C22H30N4O4S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0475480
|
6-chloro-2-oxo-N-((1R,3r,5S)-8-((piperidin-4-ylmethyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)indoline-5-carboxamide
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|
C22H29ClN4O4S
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0402928
|
2-oxo-N-((1R,3r,5S)-8-((piperidin-4-ylmethyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)indoline-5-carboxamide
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|
C22H30N4O4S
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0459466
|
1-methyl-2-oxo-N-((1R,3r,5S)-8-((piperidin-4-ylmethyl)sulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)indoline-5-carboxamide
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|
C23H32N4O4S
|
1
|
| 1 |
IC50 = 3900 nM
|
|
|
|
CP0561879
|
N-(1-((3-aminopropyl)sulfonyl)piperidin-4-yl)-6-chloro-2-oxoindoline-5-carboxamide
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|
C17H23ClN4O4S
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0383127
|
N-(1-((3-aminopropyl)sulfonyl)piperidin-4-yl)-2-oxoindoline-5-carboxamide
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|
C17H24N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0475481
|
2-oxo-N-(1-((piperidin-4-ylmethyl)sulfonyl)piperidin-4-yl)indoline-5-carboxamide
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|
C20H28N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0561880
|
2-oxo-N-(piperidin-4-yl)indoline-5-carboxamide
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|
C14H17N3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
