Brief Information of the Cell Line and Protein
Cell Line ID: CL000196 , MDA-MB-468
Synonyms
MDA-MB 468
MDA-MB468
MDAMB468
MDA-468
MDA468
MB468
MD Anderson-Metastatic Breast-468
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0419
Protein ID: PT01221 , TGF-beta receptor type-1
Gene Name TGFBR1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P36897
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000196  Protein ID: PT01221
 
Compound ID Compound Name Compound Formula
CP0472008
4-pyridinoxy-2-anilinopyridine-based compound, 5
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C25H24N4O4
 1
1
IC50 = 20 nM
   TI
   LI
   LO
   TS
CP0461213
4-pyridinoxy-2-anilinopyridine-based compound, 6
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C21H23N3O4
 1
1
IC50 = 21 nM
   TI
   LI
   LO
   TS
CP0461212
4-pyridinoxy-2-anilinopyridine-based compound, 19
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C18H18N4O3S
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS
CP0431006
4-pyridinoxy-2-anilinopyridine-based compound, 16
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C23H21N5O3S
 1
1
IC50 = 27 nM
   TI
   LI
   LO
   TS
CP0388400
4-pyridinoxy-2-anilinopyridine-based compound, 17
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C26H25N5O2
 1
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
CP0502843
4-pyridinoxy-2-anilinopyridine-based compound, 12
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C24H22N4O2
 1
1
IC50 = 32 nM
   TI
   LI
   LO
   TS
CP0418629
4-pyridinoxy-2-anilinopyridine-based compound, 14
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C24H22N4O2
 1
1
IC50 = 35 nM
   TI
   LI
   LO
   TS
CP0536658
4-pyridinoxy-2-anilinopyridine-based compound, 1
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C26H26N4O4
 1
1
IC50 = 55 nM
   TI
   LI
   LO
   TS
CP0502883
4-pyridinoxy-2-anilinopyridine-based compound, 13
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C27H27N5O2
 1
1
IC50 = 62 nM
   TI
   LI
   LO
   TS
CP0499140
4-pyridinoxy-2-anilinopyridine-based compound, 18
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C23H19FN4O
 1
1
IC50 = 63 nM
   TI
   LI
   LO
   TS
CP0397204
4-pyridinoxy-2-anilinopyridine-based compound, 10
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C24H22N4O2
 1
1
IC50 = 114 nM
   TI
   LI
   LO
   TS
CP0418635
4-pyridinoxy-2-anilinopyridine-based compound, 15
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C27H27N5O2
 1
1
IC50 = 146 nM
   TI
   LI
   LO
   TS
CP0418625
4-pyridinoxy-2-anilinopyridine-based compound, 8
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C20H21N3O4
 1
1
IC50 = 282 nM
   TI
   LI
   LO
   TS
CP0401467
4-pyridinoxy-2-anilinopyridine-based compound, 9
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C20H21N3O4
 1
1
IC50 = 628 nM
   TI
   LI
   LO
   TS
CP0502882
4-pyridinoxy-2-anilinopyridine-based compound, 11
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C27H27N5O2
 1
1
IC50 > 3000 nM
   TI
   LI
   LO
   TS
CP0454218
4-pyridinoxy-2-anilinopyridine-based compound, 7
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C19H19N3O4
 1
1
IC50 > 5800 nM
   TI
   LI
   LO
   TS