Compound ID |
Compound Name |
Compound Formula |
CP0955941
|
(S)-6-(cyclopropylmethyl)-N-((S)-1-(5-(7-methoxyquinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C34H45N5O3
|
1
|
1 |
IC50 = 0.05 nM
|
|
|
CP0636220
|
(S)-N-(1-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-7-(isoxazol-3-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H28FN5O3
|
2
|
1 |
IC50 = 0.08 nM
|
|
|
2 |
IC50 = 0.1 nM
|
|
|
CP0638656
|
(S)-N-(1-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-7-(5-methylisoxazol-3-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C25H30FN5O3
|
1
|
1 |
IC50 = 0.16 nM
|
|
|
CP0138710
|
(2S)-6-(cyclopropylmethyl)-N-[(1S)-1-[5-(7-methoxy-2-methylquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C35H46N4O4
|
1
|
1 |
IC50 = 0.17 nM
|
|
|
CP0015199
|
N-[(1S)-1-[5-(2-fluorophenyl)-1,3-oxazol-2-yl]-7-(1,2-oxazol-3-yl)-7-oxoheptyl]-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H27FN4O4
|
1
|
1 |
IC50 = 0.2 nM
|
|
|
CP0678023
|
(S)-6-ethyl-N-((S)-1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C32H43N5O3
|
1
|
1 |
IC50 = 0.22 nM
|
|
|
CP0965642
|
(S)-N-((S)-1-(5-(7-methoxy-2-(pyrrolidin-1-yl)quinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-methyl-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C35H48N6O3
|
1
|
1 |
IC50 = 0.32 nM
|
|
|
CP0569672
|
(3S,6R,9R,12R)-3-[(2S)-butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone
Show/Hide
|
C34H49N5O6
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0638831
|
(S)-7-amino-7-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-1-(isoxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
1 |
IC50 = 1.4 nM
|
|
|
CP0547778
|
(2S)-6-ethyl-N-[(1S)-1-[5-(7-methoxyquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C32H42N4O4
|
1
|
1 |
IC50 < 1.5 nM
|
|
|
CP0955940
|
(S)-6-ethyl-N-((S)-1-(5-(7-methoxyquinolin-6-yl)-1H-imidazol-2-yl)-7-oxononyl)-6-azaspiro[2.5]octane-1-carboxamide
Show/Hide
|
C32H43N5O3
|
1
|
1 |
IC50 < 1.5 nM
|
|
|
CP0531517
|
(2S)-N-[(1S)-1-[5-(7-methoxyquinolin-6-yl)-1,3-oxazol-2-yl]-7-oxononyl]-6-methyl-6-azaspiro[2.5]octane-2-carboxamide
Show/Hide
|
C31H40N4O4
|
1
|
1 |
IC50 = 1.52 nM
|
|
|
CP0637739
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-7-oxononyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C27H35N5O3
|
1
|
1 |
IC50 = 2 nM
|
|
|
CP0906813
|
3-amino-2-(5-hydroxy-2-methyl-1H-indol-3-yl)-N-((S)-1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)propanamide
Show/Hide
|
C30H34N6O3
|
1
|
1 |
IC50 = 2 nM
|
|
|
CP0003911
|
(7S)-7-amino-7-[5-(2-fluorophenyl)-1,2-oxazol-3-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H20FN3O3
|
1
|
1 |
IC50 = 3.1 nM
|
|
|
CP0639103
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-oxo-7-(thiazol-2-yl)heptyl)-1-methylpiperidine-4-carboxamide
Show/Hide
|
C26H32FN5O2S
|
1
|
1 |
IC50 = 5.8 nM
|
|
|
CP0208472
|
N-(2-amino-5-thiophen-2-ylphenyl)-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C23H23N5O3S
|
1
|
1 |
IC50 = 6 nM
|
|
|
CP0638180
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-(4-methyloxazol-2-yl)-7-oxoheptyl)-1-methylpiperidine-4-carboxamide
Show/Hide
|
C27H34FN5O3
|
1
|
1 |
IC50 = 8.3 nM
|
|
|
CP0840086
|
(S)-N-(5-(2-hydroxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27N5O3S
|
1
|
1 |
IC50 = 8.9 nM
|
|
|
CP0749584
|
(S)-N-(5-(2-fluoro-6-hydroxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H26FN5O3S
|
1
|
1 |
IC50 = 9.7 nM
|
|
|
CP0461097
|
N-(2-amino-5-thiophen-3-ylphenyl)-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C23H23N5O3S
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0638655
|
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-(oxazol-2-yl)-7-oxoheptyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H28FN5O3
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0257245
|
N-[2-amino-5-(4-methylthiophen-2-yl)phenyl]-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C24H25N5O3S
|
1
|
1 |
IC50 = 14 nM
|
|
|
CP0015198
|
(7S)-7-amino-7-[1-(4-fluorophenyl)pyrazol-4-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0951200
|
3-amino-2-(5-methoxy-2-methyl-1H-indol-3-yl)-N-((S)-1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)propanamide
Show/Hide
|
C31H36N6O3
|
1
|
1 |
IC50 = 16 nM
|
|
|
CP0299806
|
N-(2-amino-5-phenylphenyl)-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C25H25N5O3
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0371187
|
N-[2-amino-5-(1-methylpyrazol-4-yl)phenyl]-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C23H25N7O3
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0371186
|
N-[2-amino-5-(4-fluorophenyl)phenyl]-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C25H24FN5O3
|
1
|
1 |
IC50 = 20 nM
|
|
|
CP0014401
|
(7S)-7-amino-7-[1-(4-fluorophenyl)pyrazol-3-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0013328
|
(7S)-7-amino-7-[2-(4-fluorophenyl)triazol-4-yl]-1-(1,2-oxazol-3-yl)heptan-1-one
Show/Hide
|
C18H20FN5O2
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0960351
|
2-(5-Hydroxy-2-methyl-1H-indol-3-yl)-N-((S)-1-(4-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)propanamide
Show/Hide
|
C30H33N5O3
|
1
|
1 |
IC50 = 37 nM
|
|
|
CP0955787
|
(S)-N-(5-(2-amino-6-fluorobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27FN6O2S
|
1
|
1 |
IC50 = 40 nM
|
|
|
CP0951201
|
2-(5-methoxy-2-methyl-1H-indol-3-yl)-N-((S)-1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)propanamide
Show/Hide
|
C31H35N5O3
|
1
|
1 |
IC50 = 47 nM
|
|
|
CP0371188
|
N-[2-amino-5-(1-methylimidazol-4-yl)phenyl]-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C23H25N7O3
|
1
|
1 |
IC50 = 51 nM
|
|
|
CP0011354
|
N-[(1S)-1-[5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl]-7-(1,2-oxazol-3-yl)-7-oxoheptyl]-1-methylazetidine-3-carboxamide
Show/Hide
|
C23H26FN5O4
|
1
|
1 |
IC50 = 51 nM
|
|
|
CP0831925
|
(S)-N-(5-(3-hydroxypicolinamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C28H26N6O3S
|
1
|
1 |
IC50 = 52 nM
|
|
|
CP0639104
|
(S)-1-methyl-N-(7-oxo-1-(4-phenyl-1H-imidazol-2-yl)-7-(pyridin-2-yl)heptyl)piperidine-4-carboxamide
Show/Hide
|
C28H35N5O2
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0639105
|
(S)-7-amino-7-(5-(2-fluorophenyl)-1H-imidazol-2-yl)-1-(oxazol-4-yl)heptan-1-one
Show/Hide
|
C19H21FN4O2
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0637596
|
(S)-7-amino-1-(5-(hydroxymethyl)oxazol-2-yl)-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)heptan-1-one
Show/Hide
|
C24H27N5O4
|
1
|
1 |
IC50 = 194 nM
|
|
|
CP0914610
|
(S)-N-(5-(2-hydroxy-5-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0638862
|
(S)-7-amino-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-1-(5-methylisoxazol-4-yl)heptan-1-one
Show/Hide
|
C24H27N5O3
|
1
|
1 |
IC50 = 207 nM
|
|
|
CP0638821
|
(S)-7-amino-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-1-(1H-pyrazol-3-yl)heptan-1-one
Show/Hide
|
C23H26N6O2
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0914177
|
(S)-2-(5-methoxy-1H-indol-3-yl)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)acetamide
Show/Hide
|
C29H31N5O3
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0960834
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C23H29N5O2
|
1
|
1 |
IC50 = 280 nM
|
|
|
CP0951203
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)butyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C22H27N5O2
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0208474
|
N-(2-aminophenyl)-6-(2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide
Show/Hide
|
C19H21N5O3
|
1
|
1 |
IC50 = 580 nM
|
|
|
CP0951199
|
(S)-2-(1H-indol-3-yl)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)pentyl)acetamide
Show/Hide
|
C28H29N5O2
|
1
|
1 |
IC50 = 770 nM
|
|
|
CP0749709
|
(S)-N-(5-(2-hydroxy-4-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
1 |
IC50 = 800 nM
|
|
|
CP0568450
|
(7S)-7-[[2-(5-cyanoindol-1-yl)acetyl]amino]-7-[5-[4-[(dimethylamino)methyl]phenyl]-1,3-oxazol-2-yl]-N-methylheptanamide
Show/Hide
|
C31H36N6O3
|
1
|
1 |
IC50 = 1300 nM
|
|
|
CP0637595
|
(S)-7-amino-1-(1H-imidazol-2-yl)-7-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)heptan-1-one
Show/Hide
|
C23H26N6O2
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0951202
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)hexyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C24H31N5O2
|
1
|
1 |
IC50 = 4700 nM
|
|
|
CP0961838
|
(S)-N-(5-(2-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O3S
|
1
|
1 |
IC50 = 6600 nM
|
|
|
CP0835239
|
(S)-N-(5-(2-(methylamino)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H30N6O2S
|
1
|
1 |
IC50 = 15000 nM
|
|
|
CP0902876
|
(S)-N-(5-(2-mercaptobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H27N5O2S2
|
1
|
1 |
IC50 = 15000 nM
|
|
|
CP0906814
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)nonyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C27H37N5O2
|
1
|
1 |
IC50 = 18000 nM
|
|
|
CP0742396
|
(S)-N-(5-(2-(methylthio)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O2S2
|
1
|
1 |
IC50 = 20000 nM
|
|
|
CP0965923
|
(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)propyl)-1-methylazetidine-3-carboxamide
Show/Hide
|
C21H25N5O2
|
1
|
1 |
IC50 = 23000 nM
|
|
|
CP0902996
|
(S)-N-(5-(2-(dimethylamino)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H32N6O2S
|
1
|
1 |
IC50 = 25000 nM
|
|
|
CP0902998
|
N-((1S)-5-(2-(methylsulfinyl)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O3S2
|
1
|
1 |
IC50 = 25000 nM
|
|
|
CP0955788
|
(S)-N-(5-(2-cyclopropylbenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C32H31N5O2S
|
1
|
1 |
IC50 = 25000 nM
|
|
|
CP0946826
|
(S)-N-(5-(2-(1H-pyrrol-1-yl)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C33H30N6O2S
|
1
|
1 |
IC50 = 26000 nM
|
|
|
CP0552593
|
US10301323, Compound D1
Show/Hide
|
C21H20N4O
|
1
|
1 |
IC50 = 28000 nM
|
|
|
CP0914609
|
(S)-N-(5-(2-fluoro-6-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H28FN5O3S
|
1
|
1 |
IC50 = 29000 nM
|
|
|
CP0565121
|
N-[[5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl]methyl]-1-methylazetidine-3-carboxamide
Show/Hide
|
C19H21N5O2
|
1
|
1 |
IC50 = 41000 nM
|
|
|
CP0350774
|
N-[(1S)-1-[5-(2-methoxyquinolin-3-yl)-1,3,4-oxadiazol-2-yl]-5-[(2-methylsulfanylbenzoyl)amino]pentyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C29H28N6O4S2
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0767213
|
(S)-N-(5-(2-hydroxy-3-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0840085
|
(S)-N-(5-(3-aminopicolinamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C28H27N7O2S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0882461
|
(S)-N-(1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)-5-(2-(trifluoromethoxy)benzamido)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H26F3N5O3S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0882462
|
(S)-N-(1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)-5-(2-(2,2,2-trifluoroethoxy)benzamido)pentyl)thiazole-5-carboxamide
Show/Hide
|
C31H28F3N5O3S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0882463
|
(S)-N-(5-(2-cyanobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H26N6O2S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0898602
|
(S)-N-(5-(2-hydroxy-6-methoxybenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C30H29N5O4S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0902997
|
(S)-N-(5-(2-chlorobenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
Show/Hide
|
C29H26ClN5O2S
|
1
|
1 |
IC50 > 45000 nM
|
|
|
CP0928234
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(S)-N-(5-(2,3-dihydro-1H-indene-4-carboxamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
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C32H31N5O2S
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1
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1 |
IC50 > 45000 nM
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CP0928238
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(S)-N-(5-(2-(ethylthio)benzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
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C31H31N5O2S2
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1
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1 |
IC50 > 45000 nM
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CP0942943
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(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)-5-(2-(methylthio)benzamido)pentyl)thiazole-5-carboxamide
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C30H30N6O3S2
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1
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1 |
IC50 > 45000 nM
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CP0958717
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(S)-N-(5-(2-ethylbenzamido)-1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)pentyl)thiazole-5-carboxamide
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C31H31N5O2S
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1
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1 |
IC50 > 45000 nM
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CP0962479
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(S)-N-(1-(5-(2-methoxyquinolin-3-yl)-1H-imidazol-2-yl)ethyl)-1-methylazetidine-3-carboxamide
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C20H23N5O2
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1
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1 |
IC50 > 50000 nM
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