| Compound ID |
Compound Name |
Compound Formula |
|
CP0004075
|
(1S,3R)-3-acetamido-N-[5-chloro-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamide
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|
C22H28ClN5O2
|
1
|
| 1 |
EC50 = 13.7 nM
|
|
|
|
CP0004074
|
US10717746, Example 48
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|
C21H26ClN5O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0008245
|
US10717746, Example 51
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|
C23H30FN5O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0009105
|
US10717746, Example 25
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|
C22H28FN5O2
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0014318
|
US10717746, Example 27
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|
C18H21ClN4O2
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0012933
|
US10717746, Example 44
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|
C23H31N5O2
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0008759
|
US10717746, Example 22
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|
C22H28ClN5O2
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
|
CP0012360
|
US10717746, Example 47
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|
C23H31N5O2
|
1
|
| 1 |
EC50 = 74 nM
|
|
|
|
CP0013321
|
US10717746, Example 16
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|
C22H29N5O2
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0008422
|
US10717746, Example 2
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|
C21H26ClN5O2
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0011527
|
US10717746, Example 39
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|
C23H28N6O2
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0014394
|
(1S,3R)-3-acetamido-N-(5-chloro-4-pyrazolo[1,5-a]pyridin-3-ylpyridin-2-yl)cyclohexane-1-carboxamide
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|
C21H22ClN5O2
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0013322
|
US10717746, Example 63
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|
C21H26FN5O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0014392
|
US10717746, Example 66
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|
C22H28ClN5O2
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0002333
|
US9067888, 33
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|
C21H24FN3O3
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0011851
|
US10717746, Example 8
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|
C20H24ClN5O3
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0013657
|
US10717746, Example 10
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|
C20H24ClN5O2
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0013359
|
US10717746, Example 43
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|
C22H28ClN5O2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0013360
|
US10717746, Example 3
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|
C21H27N5O2
|
1
|
| 1 |
EC50 = 440 nM
|
|
|
|
CP0011852
|
(1S,3R)-3-acetamido-N-[5-chloro-4-(1,5-dimethylpyrazol-4-yl)pyridin-2-yl]cyclohexane-1-carboxamide
Show/Hide
|
C19H24ClN5O2
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0011529
|
(1S,3R)-3-acetamido-N-[4-(2-methyl-3-propan-2-ylimidazol-4-yl)pyridin-2-yl]cyclohexane-1-carboxamide
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|
C21H29N5O2
|
1
|
| 1 |
EC50 = 660 nM
|
|
|
|
CP0009290
|
US10717746, Example 15
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|
C20H25ClN6O2
|
1
|
| 1 |
EC50 = 670 nM
|
|
|
|
CP0011528
|
US10717746, Example 12
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|
C20H24ClN5O2
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0012361
|
US10717746, Example 13
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|
C21H27ClN6O2
|
1
|
| 1 |
EC50 = 910 nM
|
|
|
|
CP0012362
|
US10717746, Example 7
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|
C21H26ClN5O2
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0013261
|
US10717746, Example 11
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|
C20H24ClN5O3
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
