| Compound ID |
Compound Name |
Compound Formula |
|
CP0468707
|
2-[5-(2-chloro-4-hydroxyphenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H18ClNO4
|
2
|
| 1 |
EC50 = 9 nM
|
|
|
| 2 |
IC50 = 76 nM
|
|
|
|
CP0512850
|
2-[5-(2-fluorophenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H18FNO3
|
2
|
| 1 |
EC50 = 36 nM
|
|
|
| 2 |
IC50 = 67 nM
|
|
|
|
CP0448922
|
2-[3-[4-(4-hydroxyphenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
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|
C22H23NO4
|
2
|
| 1 |
EC50 = 70 nM
|
|
|
| 2 |
IC50 = 21 nM
|
|
|
|
CP0463250
|
2-[5-(2-fluoro-4-hydroxyphenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H18FNO4
|
2
|
| 1 |
EC50 = 80 nM
|
|
|
| 2 |
IC50 = 28 nM
|
|
|
|
CP0475369
|
2-[[(E)-5-(2-fluoro-4-hydroxyphenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
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|
C18H16FNO4
|
2
|
| 1 |
EC50 = 110 nM
|
|
|
| 2 |
IC50 = 331 nM
|
|
|
|
CP0460366
|
2-[[(E)-5-(4-hydroxyphenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
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|
C18H17NO4
|
2
|
| 1 |
EC50 = 130 nM
|
|
|
| 2 |
IC50 = 25 nM
|
|
|
|
CP0534188
|
2-[3-[4-(2-chlorophenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
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|
C22H22ClNO3
|
2
|
| 1 |
EC50 = 130 nM
|
|
|
| 2 |
IC50 = 75 nM
|
|
|
|
CP0489055
|
2-[5-(4-hydroxyphenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H19NO4
|
2
|
| 1 |
EC50 = 160 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
|
CP0460364
|
2-[5-(2-chlorophenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H18ClNO3
|
2
|
| 1 |
EC50 = 190 nM
|
|
|
| 2 |
IC50 = 56 nM
|
|
|
|
CP0474982
|
2-[3-[4-(2-fluorophenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C22H22FNO3
|
2
|
| 1 |
EC50 = 190 nM
|
|
|
| 2 |
IC50 = 282 nM
|
|
|
|
CP0512852
|
2-[3-[4-(3-hydroxyphenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
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|
C22H23NO4
|
2
|
| 1 |
EC50 = 230 nM
|
|
|
| 2 |
IC50 = 32 nM
|
|
|
|
CP0463252
|
2-[[(E)-5-(2-hydroxyphenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
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|
C18H17NO4
|
2
|
| 1 |
EC50 = 250 nM
|
|
|
| 2 |
IC50 = 37 nM
|
|
|
|
CP0482546
|
2-[3-[4-(2-fluoro-4-hydroxyphenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C22H22FNO4
|
2
|
| 1 |
EC50 = 260 nM
|
|
|
| 2 |
IC50 = 58 nM
|
|
|
|
CP0474978
|
2-[[(E)-5-(2-chlorophenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
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|
C18H16ClNO3
|
2
|
| 1 |
EC50 = 270 nM
|
|
|
| 2 |
IC50 = 88 nM
|
|
|
|
CP0512854
|
2-[[(E)-5-(3-hydroxyphenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H17NO4
|
2
|
| 1 |
EC50 = 390 nM
|
|
|
| 2 |
IC50 = 383 nM
|
|
|
|
CP0515604
|
2-[3-[4-(2-hydroxyphenyl)phenyl]propanoylamino]cyclohexene-1-carboxylic acid
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|
C22H23NO4
|
2
|
| 1 |
EC50 = 410 nM
|
|
|
| 2 |
IC50 = 40 nM
|
|
|
|
CP0463251
|
2-[[(E)-5-(2-fluorophenyl)pent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H16FNO3
|
2
|
| 1 |
EC50 = 450 nM
|
|
|
| 2 |
IC50 = 16 nM
|
|
|
|
CP0489056
|
2-[5-(4-fluorophenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C18H18FNO3
|
2
|
| 1 |
EC50 = 630 nM
|
|
|
| 2 |
IC50 = 291 nM
|
|
|
|
CP0512851
|
2-[5-(2-hydroxyphenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H19NO4
|
2
|
| 1 |
EC50 = 720 nM
|
|
|
| 2 |
IC50 = 229 nM
|
|
|
|
CP0389419
|
2-[3-(6-hydroxynaphthalen-2-yl)prop-2-ynoylamino]cyclohexene-1-carboxylic acid
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|
C20H17NO4
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0384489
|
2-[[(E)-5-phenylpent-2-en-4-ynoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H17NO3
|
3
|
| 1 |
EC50 = 1010 nM
|
|
|
| 2 |
EC50 = 3600 nM
|
|
|
| 3 |
IC50 = 327 nM
|
|
|
|
CP0471407
|
2-[[(E)-3-(6-hydroxynaphthalen-2-yl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C20H19NO4
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0384940
|
2-(3-(6-hydroxynaphthalen-2-yl)propanamido)cyclohex-1-enecarboxylic acid
Show/Hide
|
C20H21NO4
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
|
CP0512853
|
2-[5-(3-hydroxyphenyl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H19NO4
|
2
|
| 1 |
EC50 = 2980 nM
|
|
|
| 2 |
IC50 = 138 nM
|
|
|
|
CP0463249
|
2-[5-(5-hydroxypyridin-2-yl)pent-4-ynoylamino]cyclohexene-1-carboxylic acid
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|
C17H18N2O4
|
2
|
| 1 |
EC50 = 3370 nM
|
|
|
| 2 |
IC50 = 665 nM
|
|
|
|
CP0384941
|
2-[[(E)-3-quinolin-2-ylprop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C19H18N2O3
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0389441
|
2-[3-(2-chloro-6-methoxyquinolin-3-yl)propanoylamino]cyclohexene-1-carboxylic acid
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|
C20H21ClN2O4
|
1
|
| 1 |
EC50 = 4100 nM
|
|
|
|
CP0427232
|
2-[[(E)-3-naphthalen-2-ylprop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C20H19NO3
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0534187
|
4-[5-[(2-carboxycyclohexen-1-yl)amino]-5-oxopent-1-ynyl]benzoic acid
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|
C19H19NO5
|
2
|
| 1 |
EC50 = 5610 nM
|
|
|
| 2 |
IC50 = 3620 nM
|
|
|
|
CP0400828
|
2-[[(E)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C17H17NO5
|
1
|
| 1 |
EC50 = 5800 nM
|
|
|
|
CP0469009
|
2-[[(E)-3-(2-chloro-6-methoxyquinolin-3-yl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C20H19ClN2O4
|
1
|
| 1 |
EC50 = 6300 nM
|
|
|
|
CP0448275
|
2-[[(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H19NO5
|
1
|
| 1 |
EC50 = 6800 nM
|
|
|
|
CP0427263
|
2-(3-naphthalen-2-ylpropanoylamino)cyclohexene-1-carboxylic acid
Show/Hide
|
C20H21NO3
|
1
|
| 1 |
EC50 = 8300 nM
|
|
|
|
CP0427231
|
2-[[(1R,2R)-2-naphthalen-2-ylcyclopropanecarbonyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
EC50 = 12500 nM
|
|
|
|
CP0482541
|
2-[[(E)-5-phenylpent-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H21NO3
|
2
|
| 1 |
EC50 = 19600 nM
|
|
|
| 2 |
IC50 = 2828 nM
|
|
|
|
CP0384487
|
2-[[(E)-3-(2-chloro-3,4-dimethoxyphenyl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C18H20ClNO5
|
1
|
| 1 |
EC50 = 26300 nM
|
|
|
|
CP0389421
|
2-[[(E)-3-(2-chloroquinolin-3-yl)prop-2-enoyl]amino]cyclohexene-1-carboxylic acid
Show/Hide
|
C19H17ClN2O3
|
1
|
| 1 |
EC50 = 27400 nM
|
|
|
|
CP0384490
|
2-[3-(2-methylquinolin-6-yl)propanoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C20H22N2O3
|
1
|
| 1 |
EC50 = 36400 nM
|
|
|
|
CP0469008
|
2-[3-(1,3-benzodioxol-5-yl)propanoylamino]cyclohexene-1-carboxylic acid
Show/Hide
|
C17H19NO5
|
1
|
| 1 |
EC50 = 51600 nM
|
|
|
