| Compound ID |
Compound Name |
Compound Formula |
|
CP0236110
|
2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-[(2R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethoxy)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]pyridine-3-carboxamide
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|
C30H30ClF3N4O6
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
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CP0075555
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N-[(1R,2S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]nonanamide
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|
C24H38N2O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0091328
|
2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxo-3-phenylmethoxypropan-2-yl]pyridine-3-carboxamide
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|
C28H28ClF3N4O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0191300
|
N-[(1R,2S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-hydroxy-3-pyrrolidin-1-ylpropan-2-yl]octanamide
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|
C23H36N2O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0368789
|
N-[(2S)-1-[(1R,5S)-3-amino-8-azabicyclo[3.2.1]octan-8-yl]-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl]-1-(2,4-dichlorophenyl)cyclopropane-1-carboxamide
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|
C26H27Cl4N3O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0443642
|
N-[(2S)-3-(4-chlorophenyl)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-1-(2,4-dichlorophenyl)cyclopropane-1-carboxamide
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|
C24H26Cl3N3O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0075556
|
N-[(2R)-1-[[(3S)-1-azabicyclo[2.2.2]octan-3-yl]amino]-1-oxo-3-phenylmethoxypropan-2-yl]-2-[2-chloro-4-(trifluoromethyl)phenoxy]pyridine-3-carboxamide
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|
C30H30ClF3N4O4
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0443643
|
1-(2,4-dichlorophenyl)-N-[(2S)-3-(2,4-dichlorophenyl)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]cyclopropane-1-carboxamide
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|
C24H25Cl4N3O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
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CP0070455
|
2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-[(2R)-1-[(3R)-3-(methylamino)pyrrolidin-1-yl]-1-oxo-3-phenylmethoxypropan-2-yl]pyridine-3-carboxamide
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|
C28H28ClF3N4O4
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0057863
|
1-(2,4-dichlorophenyl)-N-[(2S)-3-(1H-indol-3-yl)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]cyclopropane-1-carboxamide
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|
C26H28Cl2N4O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0057860
|
N-[(2S)-1-[(1S,5R)-3-amino-8-azabicyclo[3.2.1]octan-8-yl]-3-(2,4-dichlorophenyl)-1-oxopropan-2-yl]-1-[4-(trifluoromethoxy)phenyl]cyclopropane-1-carboxamide
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|
C27H28Cl2F3N3O3
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0413929
|
N-[(2S)-3-(4-bromophenyl)-1-[2-(dimethylamino)ethyl-methylamino]-1-oxopropan-2-yl]-1-(2,4-dichlorophenyl)cyclopropane-1-carboxamide
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|
C24H28BrCl2N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
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CP0264143
|
N-[(2R)-1-[[(3R)-1-azabicyclo[2.2.2]octan-3-yl]amino]-1-oxo-3-phenylmethoxypropan-2-yl]-2-[2-chloro-4-(trifluoromethyl)phenoxy]pyridine-3-carboxamide
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|
C30H30ClF3N4O4
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0084536
|
2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-[(2R)-3-[(4-fluorophenyl)methoxy]-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]pyridine-3-carboxamide
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|
C28H27ClF4N4O4
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
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CP0046329
|
N-[(2S)-3-(4-bromophenyl)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-1-(2,4-dichlorophenyl)cyclopropane-1-carboxamide
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|
C24H26BrCl2N3O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0086232
|
N-[(2S)-1-[(1S,5R)-3-amino-8-azabicyclo[3.2.1]octan-8-yl]-3-(4-bromophenyl)-1-oxopropan-2-yl]-1-[4-(trifluoromethoxy)phenyl]cyclopropane-1-carboxamide
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|
C27H29BrF3N3O3
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
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CP0356015
|
N-[(2S)-1-[(1R,5S)-3-amino-8-azabicyclo[3.2.1]octan-8-yl]-3-(4-bromophenyl)-1-oxopropan-2-yl]-1-(2,4-dichlorophenyl)cyclopropane-1-carboxamide
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|
C26H28BrCl2N3O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
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CP0210742
|
2-[2-chloro-4-(trifluoromethyl)phenoxy]-N-[(2R)-3-[(2-methyl-1,3-oxazol-5-yl)methoxy]-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]pyridine-3-carboxamide
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|
C26H27ClF3N5O5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
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CP0565817
|
1-(2,4-dichlorophenyl)-N-[(2S)-3-(2,4-dichlorophenyl)-1-[2-(dimethylamino)ethyl-methylamino]-1-oxopropan-2-yl]cyclopropane-1-carboxamide
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|
C24H27Cl4N3O2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0120672
|
1-(2,4-dichlorophenyl)-N-[(2S)-1-(4-methylpiperazin-1-yl)-1-oxo-3-phenylmethoxypropan-2-yl]cyclopropane-1-carboxamide
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|
C25H29Cl2N3O3
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
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CP0045196
|
(2R,3R,4R,5S)-1-[5-(Adamantan-1-ylmethoxy)-pentyl]-2-hydroxymethyl-piperidine-3,4,5-triol
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|
C22H39NO5
|
1
|
| 1 |
IC50 = 16500 nM
|
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