Brief Information of the Cell Line and Protein
Cell Line ID: CL000068 , A-549
Synonyms
A 549
A549
NCI-A549
A549/ATCC
A549 ATCC
A549ATCC
hA549
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0023
Protein ID: PT00825 , 5-hydroxytryptamine receptor 2A
Gene Name HTR2A
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P28223
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000068  Protein ID: PT00825
 
Compound ID Compound Name Compound Formula
CP0677987
N-(2-[3H-OCH3]benzyl)-2-(2-[3H-OCH3]-5-methoxy-4-iodophenyl)ethylamine
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C18H22INO3
 1
1
Kd = 0.097 nM
   TI
   LI
   LO
   TS
CP0896941
[3H]-3-(2-(4-(4-fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione
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C22H22FN3O3
 1
1
Kd = 2.2 nM
   TI
   LI
   LO
   TS
CP0045725
(4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[7.6.1.0^{2,7}.0^{12,16}]hexadeca-1(16),2,9,12,14-pentaene-4-carboxamide
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C20H25N3O
 2
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
2
Ki = 4 nM
   TI
   LI
   LO
   TS
CP0208552
(E)-N-[2-(3-Dimethylamino-propylsulfanyl)-phenyl]-3-phenyl-acrylamide
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C20H24N2OS
 2
1
Ki = 17 nM
   TI
   LI
   LO
   TS
2
Ki = 24 nM
   TI
   LI
   LO
   TS
CP0055945
1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine
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C11H16INO2
 2
1
Ki = 28 nM
   TI
   LI
   LO
   TS
2
Ki = 29 nM
   TI
   LI
   LO
   TS
CP0001238
14C-5-hydroxy tryptamine creatinine disulfate
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C10H12N2O
 2
1
Ki = 120 nM
   TI
   LI
   LO
   TS
2
Ki = 160 nM
   TI
   LI
   LO
   TS