| Compound ID |
Compound Name |
Compound Formula |
|
CP0000305
|
(-)-(etorphine)
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|
C17H19NO3
|
1
|
| 1 |
Ki = 6.08 nM
|
|
|
|
CP0475186
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-isoquinolin-6-ylurea
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|
C32H34F3N5O
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0383002
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-quinolin-5-ylurea
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|
C32H34F3N5O
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0443798
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-[3-fluoro-4-[(sulfamoylamino)methyl]phenyl]urea
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|
C30H36F4N6O3S
|
1
|
| 1 |
Ki = 72.4 nM
|
|
|
|
CP0443801
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-[[3-fluoro-4-(methanesulfonamido)phenyl]methyl]urea
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|
C31H37F4N5O3S
|
1
|
| 1 |
Ki = 76.2 nM
|
|
|
|
CP0443799
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-(1-oxo-2H-isoquinolin-5-yl)urea
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|
C32H34F3N5O2
|
1
|
| 1 |
Ki = 105 nM
|
|
|
|
CP0468924
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-(7-hydroxynaphthalen-1-yl)urea
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|
C33H35F3N4O2
|
1
|
| 1 |
Ki = 137 nM
|
|
|
|
CP0470976
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-quinolin-7-ylurea
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|
C32H34F3N5O
|
1
|
| 1 |
Ki = 166 nM
|
|
|
|
CP0460555
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-isoquinolin-7-ylurea
Show/Hide
|
C32H34F3N5O
|
1
|
| 1 |
Ki = 177 nM
|
|
|
|
CP0470975
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-isoquinolin-8-ylurea
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|
C32H34F3N5O
|
1
|
| 1 |
Ki = 205 nM
|
|
|
|
CP0470715
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-(2,3-dihydro-1-benzofuran-6-yl)urea
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|
C31H35F3N4O2
|
1
|
| 1 |
Ki = 225 nM
|
|
|
|
CP0383001
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-(2-oxo-1H-quinolin-5-yl)urea
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|
C32H34F3N5O2
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0470972
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-[3-fluoro-4-(hydroxymethyl)phenyl]urea
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|
C30H34F4N4O2
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0470977
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-(7-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl)urea
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|
C33H39F3N4O2
|
1
|
| 1 |
Ki = 261 nM
|
|
|
|
CP0470979
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-[3-fluoro-4-(methanesulfonamidomethyl)phenyl]urea
Show/Hide
|
C31H37F4N5O3S
|
1
|
| 1 |
Ki = 322 nM
|
|
|
|
CP0437983
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-[3-fluoro-4-(methanesulfonamido)phenyl]urea
Show/Hide
|
C30H35F4N5O3S
|
1
|
| 1 |
Ki = 368 nM
|
|
|
|
CP0536351
|
N-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide
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|
C32H38F4N4O3S
|
1
|
| 1 |
Ki = 428 nM
|
|
|
|
CP0536350
|
1-[[2-[4-benzyl-4-(dimethylamino)piperidin-1-yl]-4-(trifluoromethyl)phenyl]methyl]-3-isoquinolin-5-ylurea
Show/Hide
|
C32H34F3N5O
|
1
|
| 1 |
Ki = 507 nM
|
|
|
