Compound ID |
Compound Name |
Compound Formula |
CP0105598
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-[2-(trifluoromethoxy)phenoxy]-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H15ClF3N3O2
|
1
|
1 |
IC50 = 0.5 nM
|
|
|
CP0105607
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridine
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|
C18H18ClN3
|
1
|
1 |
IC50 = 0.61 nM
|
|
|
CP0572781
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(2-fluorophenoxy)-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H15ClFN3O
|
1
|
1 |
IC50 = 0.7 nM
|
|
|
CP0053206
|
4-[2-[[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]oxy]phenyl]morpholine
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|
C25H23ClN4O2
|
1
|
1 |
IC50 = 0.9 nM
|
|
|
CP0053207
|
8-(2-chlorophenoxy)-3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H15Cl2N3O
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0353988
|
2-[[3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridin-8-yl]oxy]phenol
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|
C21H16ClN3O2
|
1
|
1 |
IC50 = 1.4 nM
|
|
|
CP0105606
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-cyclopropyl-[1,2,4]triazolo[4,3-a]pyridine
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|
C18H16ClN3
|
1
|
1 |
IC50 = 1.6 nM
|
|
|
CP0487807
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-phenoxy-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H16ClN3O
|
1
|
1 |
IC50 = 1.7 nM
|
|
|
CP0406166
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-cyclobutyl-[1,2,4]triazolo[4,3-a]pyridine
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|
C19H18ClN3
|
1
|
1 |
IC50 = 2.4 nM
|
|
|
CP0105597
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(2-phenylphenoxy)-[1,2,4]triazolo[4,3-a]pyridine
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|
C27H20ClN3O
|
1
|
1 |
IC50 = 2.7 nM
|
|
|
CP0105594
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-cyclobutyloxy-[1,2,4]triazolo[4,3-a]pyridine
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|
C19H18ClN3O
|
1
|
1 |
IC50 = 4.2 nM
|
|
|
CP0400696
|
4-[8-(2-fluorophenoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]bicyclo[2.2.1]heptan-1-ol
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|
C19H18FN3O2
|
1
|
1 |
IC50 = 5.1 nM
|
|
|
CP0105596
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(2-methylpyridin-3-yl)oxy-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H17ClN4O
|
1
|
1 |
IC50 = 5.5 nM
|
|
|
CP0547693
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(2-methylsulfonylphenoxy)-[1,2,4]triazolo[4,3-a]pyridine
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|
C22H18ClN3O3S
|
1
|
1 |
IC50 = 8.1 nM
|
|
|
CP0415507
|
3-cycloheptyl-8-[(2,6-dichlorophenoxy)methyl]-[1,2,4]triazolo[4,3-a]pyridine
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|
C20H21Cl2N3O
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0406167
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-methyl-[1,2,4]triazolo[4,3-a]pyridine
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|
C16H14ClN3
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0406165
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-naphthalen-2-yloxy-[1,2,4]triazolo[4,3-a]pyridine
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|
C25H18ClN3O
|
1
|
1 |
IC50 = 20 nM
|
|
|
CP0353986
|
8-(4-chlorophenoxy)-3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H15Cl2N3O
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0105600
|
8-(3-chlorophenoxy)-3-[1-(4-chlorophenyl)cyclopropyl]-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H15Cl2N3O
|
1
|
1 |
IC50 = 22 nM
|
|
|
CP0105604
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-cyclohexyloxy-[1,2,4]triazolo[4,3-a]pyridine
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|
C21H22ClN3O
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0368636
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(cyclopropylmethoxy)-[1,2,4]triazolo[4,3-a]pyridine
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|
C19H18ClN3O
|
1
|
1 |
IC50 = 51 nM
|
|
|
CP0258806
|
3-[1-(4-chlorophenyl)cyclopropyl]-8-(oxan-4-yloxy)-[1,2,4]triazolo[4,3-a]pyridine
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|
C20H20ClN3O2
|
1
|
1 |
IC50 = 65 nM
|
|
|