Brief Information of the Cell Line and Protein
Cell Line ID: CL000063 , Hep-G2
Synonyms
HEP-G2
Hep G2
HEP G2
HepG2
HEPG2
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0027
Protein ID: PT01201 , Hepatocyte growth factor receptor
Gene Name MET
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P08581
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000063  Protein ID: PT01201
 
Compound ID Compound Name Compound Formula
CP0079979
(2S)-2-[[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]amino]-N-(4-imidazo[2,1-b][1,3]benzothiazol-2-ylphenyl)-3-phenylpropanamide
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C34H24F6N4O2S
 1
1
IC50 = 321 nM
   TI
   LI
   LO
   TS
CP0388720
(2R)-2-[[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]amino]-N-(4-imidazo[2,1-b][1,3]benzothiazol-2-ylphenyl)-3-phenylpropanamide
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C34H24F6N4O2S
 1
1
IC50 = 620 nM
   TI
   LI
   LO
   TS
CP0023994
(3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]-1H-PYRROL-2-YL}METHYLENE)-N-METHYL-2-OXOINDOLINE-5-SULFONAMIDE
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C28H30ClN5O4S
 1
1
IC50 = 1561 nM
   TI
   LI
   LO
   TS
CP0392886
(2S)-2-[[2-(3,5-dimethylphenyl)acetyl]amino]-N-(4-imidazo[2,1-b][1,3]benzothiazol-2-ylphenyl)-3-phenylpropanamide
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C34H30N4O2S
 1
1
IC50 = 1561 nM
   TI
   LI
   LO
   TS