Compound ID |
Compound Name |
Compound Formula |
CP0543674
|
4-(3-(4-amino-5-(8-fluoro-2-phenylquinolin-7-yl)imidazo[1,5-f][1,2,4]triazin-7-yl)cyclobutyl)piperazine-1-carbaldehyde
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|
C29H27FN8O
|
1
|
1 |
IC50 = 48 nM
|
|
|
CP0465696
|
5-(8-fluoro-2-phenylquinolin-7-yl)-7-(3-(4-methylpiperazin-1-yl)cyclobutyl)imidazo[1,5-f][1,2,4]triazin-4-amine
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|
C29H29FN8
|
1
|
1 |
IC50 = 68 nM
|
|
|
CP0162376
|
3-[4-amino-5-(8-fluoro-2-phenylquinolin-7-yl)imidazo[5,1-f][1,2,4]triazin-7-yl]-1-methylcyclobutan-1-ol
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|
C25H21FN6O
|
1
|
1 |
IC50 = 76 nM
|
|
|
CP0503936
|
4-(3-(4-amino-5-(2-phenylquinolin-7-yl)imidazo[1,5-f][1,2,4]triazin-7-yl)cyclobutyl)piperazine-1-carbaldehyde
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|
C29H28N8O
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0487314
|
7-(3-(4-methylpiperazin-1-yl)cyclobutyl)-5-(2-phenylquinolin-7-yl)imidazo[1,5-f][1,2,4]triazin-4-amine
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|
C29H30N8
|
1
|
1 |
IC50 = 320 nM
|
|
|
CP0510127
|
3-[4-amino-5-(2-phenylquinolin-7-yl)imidazo[5,1-f][1,2,4]triazin-7-yl]-1-methylcyclobutan-1-ol
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|
C25H22N6O
|
1
|
1 |
IC50 = 700 nM
|
|
|
CP0011819
|
4-(3,4-Dimethoxy-phenoxy)-6,7-dimethoxy-quinoline
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|
C19H19NO5
|
1
|
1 |
IC50 > 100000 nM
|
|
|