Brief Information of the Cell Line and Protein
Cell Line ID: CL000063 , Hep-G2
Synonyms
HEP-G2
Hep G2
HEP G2
HepG2
HEPG2
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0027
Protein ID: PT00959 , Ribosomal protein S6 kinase alpha-1
Gene Name RPS6KA1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID Q15418
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000063  Protein ID: PT00959
 
Compound ID Compound Name Compound Formula
CP0500919
US9388171, II-64
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C27H30N6O2
 1
1
IC50 = 5.47 nM
   TI
   LI
   LO
   TS
CP0564085
US9388171, I-6
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C24H27FN4O3
 1
1
IC50 = 5.96 nM
   TI
   LI
   LO
   TS
CP0515120
US9388171, II-2
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C24H25ClFN3O2
 1
1
IC50 = 8.5 nM
   TI
   LI
   LO
   TS
CP0324959
US9388171, I-8
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C21H18ClFN6O2
 1
1
IC50 = 9.84 nM
   TI
   LI
   LO
   TS
CP0324711
US9388171, II-15
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C25H21ClFN7O
 1
1
IC50 = 9.97 nM
   TI
   LI
   LO
   TS
CP0324712
US9388171, II-12
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C23H23ClFN3O3
 1
1
IC50 = 14.8 nM
   TI
   LI
   LO
   TS
CP0274071
US9388171, II-46
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C24H23ClFN5O
 1
1
IC50 = 15.7 nM
   TI
   LI
   LO
   TS
CP0483378
US9388171, I-5
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C22H22ClFN4O3
 1
1
IC50 = 16.3 nM
   TI
   LI
   LO
   TS
CP0340458
US9388171, I-21
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C26H27FN6O3
 1
1
IC50 = 18.7 nM
   TI
   LI
   LO
   TS
CP0269483
US9388171, II-37
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C27H26FN7O2
 1
1
IC50 = 30.4 nM
   TI
   LI
   LO
   TS
CP0241393
US9388171, I-24
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C24H25FN6O3
 1
1
IC50 = 37.8 nM
   TI
   LI
   LO
   TS
CP0823713
US9388171, II-23
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C22H21FN4O2
 1
1
IC50 = 65.1 nM
   TI
   LI
   LO
   TS
CP0273971
US9388171, I-11
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C21H20ClFN4O2
 1
1
IC50 = 98.9 nM
   TI
   LI
   LO
   TS
CP0324960
US9388171, I-30
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C22H22ClFN4O2
 1
1
IC50 = 476 nM
   TI
   LI
   LO
   TS