| Compound ID |
Compound Name |
Compound Formula |
|
CP0038839
|
(4R,4aS,7aR,12bS)-3-allyl-4a,9-dihydroxy-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-one;hydrochloride
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|
C19H21NO4
|
1
|
| 1 |
Kd = 3 nM
|
|
|
|
CP0402338
|
8-Cycloundecyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C24H37N3O
|
1
|
| 1 |
Ki = 0.21 nM
|
|
|
|
CP0431654
|
8-Cyclododecyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C25H39N3O
|
1
|
| 1 |
Ki = 0.28 nM
|
|
|
|
CP0422910
|
8-Cyclodecyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C23H35N3O
|
1
|
| 1 |
Ki = 0.66 nM
|
|
|
|
CP0402390
|
8-Bicyclohexyl-4-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C25H37N3O
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0405159
|
8-Cyclononyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C22H33N3O
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0437276
|
8-(4-Isopropyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C22H33N3O
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0038465
|
8-(R)-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C25H25N3O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0414949
|
8-(4-tert-Butyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C23H35N3O
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0405179
|
1-Phenyl-8-(4-propyl-cyclohexyl)-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C22H33N3O
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
|
CP0460264
|
8-(4-Isopropyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C22H33N3O
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0441527
|
8-Cyclooctyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C21H31N3O
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0422928
|
8-Cycloheptyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C20H29N3O
|
1
|
| 1 |
Ki = 51 nM
|
|
|
|
CP0379320
|
8-(4-Methyl-cyclohexyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C20H29N3O
|
1
|
| 1 |
Ki = 64 nM
|
|
|
|
CP0402183
|
8-Cyclohexyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
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|
C19H27N3O
|
1
|
| 1 |
Ki = 158 nM
|
|
|