Brief Information of the Cell Line and Protein
Cell Line ID: CL000051 , BHK-21
Synonyms
BHK 21
BHK21
Baby Hamster Kidney-21
Baby Hamster Kidney 21
Baby Hamster Kidney from litter No. 21
BHK
Category Spontaneously immortalized cell line
Organism
Mesocricetus auratus (Golden hamster)
Cellosaurus ID
CVCL_1914
Protein ID: PT01156 , Muscarinic acetylcholine receptor M4
Gene Name CHRM4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P08173
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000051  Protein ID: PT01156
 
Compound ID Compound Name Compound Formula
CP0371787
5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine; oxalic acid
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C14H23N3OS
 2
1
EC50 = 6.2 nM
   TI
   LI
   LO
   TS
2
Ki = 72 nM
   TI
   LI
   LO
   TS
CP0000324
2-acetoxyethyl(trimethyl)ammonium;bromide
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C7H16NO2+
 1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CP0377069
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-(3,4-dimethoxyphenyl)acetamide
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C27H33F2N3O4
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0128076
8-Chloro-11-piperazin-1-yl-5H-dibenzo[b,e][1,4]diazepine
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C17H17ClN4
 2
1
EC50 = 400 nM
   TI
   LI
   LO
   TS
2
Ki = 290 nM
   TI
   LI
   LO
   TS
CP0109931
ATROPEN
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C17H23NO3
 1
1
Ki = 3 nM
   TI
   LI
   LO
   TS
CP0305211
1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
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C25H32N4O
 1
1
Ki = 130 nM
   TI
   LI
   LO
   TS
CP0029624
4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one
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C20H31NO
 1
1
Ki = 1400 nM
   TI
   LI
   LO
   TS
CP0026924
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide
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C24H29N3O3
 1
1
Ki = 6900 nM
   TI
   LI
   LO
   TS