Brief Information of the Cell Line and Protein
Cell Line ID: CL000050 , HEK293-A
Synonyms
HEK-293A
HEK293A
HEK 293A
293A
QBI-HEK 293A
QBI-293A
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_6910
Protein ID: PT01279 , Adenosine receptor A3
Gene Name ADORA3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P0DMS8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000050  Protein ID: PT01279
 
Compound ID Compound Name Compound Formula
CP0534879
1-N-[3-[8-(1-adamantyl)-2,6-dioxo-1-propyl-7H-purin-3-yl]propyl]-4-N-[2-[3-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propanoylamino]ethyl]benzene-1,4-dicarboxamide
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C63H72BF2N11O8S
 1
1
Kd = 58.88 nM
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CP0534878
N-[2-[3-[3-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propanoylamino]propanoylamino]ethyl]-4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)bicyclo[2.2.2]octane-1-carboxamide
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C57H70BF2N11O8S
 1
1
Kd = 134.9 nM
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CP0534877
(2E)-1-[6-[[3-[[3-[2-[[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)bicyclo[2.2.2]octane-1-carbonyl]amino]ethylamino]-3-oxopropyl]amino]-3-oxopropyl]amino]-6-oxohexyl]-3,3-dimethyl-2-[(2E,4E)-5-(1,3,3-trimethyl-5-sulfoindol-1-ium-2-yl)penta-2,4-dienylidene]indole-5-sulfonate
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C60H80N10O12S2
 1
1
Kd > 1000 nM
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