Brief Information of the Cell Line and Protein
Cell Line ID: CL000050 , HEK293-A
 Cell Line Info 
Synonyms
HEK-293A
HEK293A
HEK 293A
293A
QBI-HEK 293A
QBI-293A
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_6910
Protein ID: PT00840 , Adenosine receptor A1
 Protein Info 
Gene Name ADORA1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P30542
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000050
 Cell Line Info 
 Protein ID: PT00840
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0534878
 Compound Info 
N-[2-[3-[3-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propanoylamino]propanoylamino]ethyl]-4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)bicyclo[2.2.2]octane-1-carboxamide
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C57H70BF2N11O8S
  2
1
Kd = 1.175 nM
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2
Kd = 3.09 nM
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CP0534879
 Compound Info 
1-N-[3-[8-(1-adamantyl)-2,6-dioxo-1-propyl-7H-purin-3-yl]propyl]-4-N-[2-[3-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propanoylamino]ethyl]benzene-1,4-dicarboxamide
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C63H72BF2N11O8S
  5
1
Kd = 3.162 nM
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2
Kd = 13.18 nM
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3
Ki = 1.413 nM
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4
Ki = 20.89 nM
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5
Ki = 1096.48 nM
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CP0534877
 Compound Info 
(2E)-1-[6-[[3-[[3-[2-[[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)bicyclo[2.2.2]octane-1-carbonyl]amino]ethylamino]-3-oxopropyl]amino]-3-oxopropyl]amino]-6-oxohexyl]-3,3-dimethyl-2-[(2E,4E)-5-(1,3,3-trimethyl-5-sulfoindol-1-ium-2-yl)penta-2,4-dienylidene]indole-5-sulfonate
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C60H80N10O12S2
  5
1
Kd = 44.67 nM
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2
Kd = 138.04 nM
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3
Ki = 0.7079 nM
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4
Ki = 7.413 nM
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5
Ki = 398.11 nM
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