| Compound ID |
Compound Name |
Compound Formula |
|
CP0095953
|
ENZALUTAMIDE
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|
C21H16F4N4O2S
|
2
|
| 1 |
EC50 = 1070 nM
|
|
|
| 2 |
EC50 = 11390 nM
|
|
|
|
CP0499654
|
US9428460, 23
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|
C23H20FN3O2
|
3
|
| 1 |
IC50 = 9 nM
|
|
|
| 2 |
IC50 = 30 nM
|
|
|
| 3 |
IC50 = 52 nM
|
|
|
|
CP0492626
|
US9428460, 24
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|
C23H19F2N3O2
|
3
|
| 1 |
IC50 = 14 nM
|
|
|
| 2 |
IC50 = 72 nM
|
|
|
| 3 |
IC50 = 92 nM
|
|
|
|
CP0489543
|
US9428460, 26
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|
C21H20N4O3
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0497655
|
US9428460, 2
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|
C20H20BrN3O3
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0444911
|
US9428460, 19
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|
C22H21FN2O2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0545344
|
N-[(2R)-1-[3-(3-chloro-4-cyanophenyl)pyrazol-1-yl]propan-2-yl]-5-(1-hydroxyethyl)-1H-pyrazole-3-carboxamide
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|
C19H19ClN6O2
|
2
|
| 1 |
IC50 = 37 nM
|
|
|
| 2 |
IC50 = 64 nM
|
|
|
|
CP0565751
|
US9428460, 30
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|
C23H19F2N3O2
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0451343
|
US9428460, 28
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|
C24H22FN3O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0515427
|
US9428460, 3
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|
C22H20F2N2O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0480876
|
US9428460, 9
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|
C23H22F2N2O2
|
3
|
| 1 |
IC50 = 56 nM
|
|
|
| 2 |
IC50 = 72 nM
|
|
|
| 3 |
IC50 = 105 nM
|
|
|
|
CP0563444
|
US9428460, 29
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|
C23H19ClFN3O2
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0480875
|
US9428460, 27
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|
C23H19ClFN3O2
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0515428
|
US9428460, 14
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|
C23H22BrFN2O2
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0545599
|
US9428460, 12
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|
C22H20BrFN2O2
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0480874
|
US9428460, 25
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|
C23H20FN3O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0480873
|
US9428460, 13
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|
C22H19BrF2N2O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0273406
|
2-[1-(3-chloro-4-cyanophenyl)pyrazol-3-yl]-N-(6-fluoropyridin-3-yl)acetamide
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|
C17H11ClFN5O
|
3
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
IC50 = 270 nM
|
|
|
| 3 |
IC50 = 460 nM
|
|
|
|
CP0451342
|
US9428460, 10
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|
C23H23FN2O2
|
3
|
| 1 |
IC50 = 175 nM
|
|
|
| 2 |
IC50 = 194 nM
|
|
|
| 3 |
IC50 = 220 nM
|
|
|
|
CP0492960
|
US9428460, 18
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|
C22H19BrClFN2O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0497656
|
US9428460, 11
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|
C21H23N3O3
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0545597
|
US9428460, 4
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|
C21H22FN3O3
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0545596
|
US9428460, 1
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|
C23H22F2N2O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0355222
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(4-fluorophenyl)acetamide
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|
C19H12F4N4O
|
2
|
| 1 |
IC50 = 250 nM
|
|
|
| 2 |
IC50 = 910 nM
|
|
|
|
CP0564112
|
US9428460, 15
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|
C23H20BrN3O2
|
1
|
| 1 |
IC50 = 261 nM
|
|
|
|
CP0572456
|
US9428460, 22
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|
C24H23N3O2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0916592
|
US9428460, 8
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|
C20H21FN4O2
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0561636
|
US9428460, 5
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|
C20H20FN3O3
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0515429
|
US9428460, 16
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|
C23H19BrF4N2O2
|
1
|
| 1 |
IC50 = 463 nM
|
|
|
|
CP0483364
|
US9428460, 17
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|
C22H20BrFN2O2
|
1
|
| 1 |
IC50 = 477 nM
|
|
|
|
CP0480872
|
US9428460, 7
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|
C21H22FN3O3
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0515430
|
US9428460, 21
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|
C20H20BrN3O3
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0565738
|
US9428460, 32
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|
C22H22N4O3
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0565737
|
US9428460, 20
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|
C21H22BrN3O3
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0451345
|
US9428460, 31
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|
C21H20N4O3
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0545598
|
US9428460, 6
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|
C20H20FN3O3
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0260233
|
2-[1-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-3-yl]-N-(6-fluoropyridin-3-yl)acetamide
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|
C18H11F4N5O
|
2
|
| 1 |
IC50 = 1120 nM
|
|
|
| 2 |
IC50 = 1310 nM
|
|
|
|
CP0386608
|
1,8-dichloro-10-[(3-hydroxy-4-methoxyphenyl)methylidene]anthracen-9-one
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|
C22H14Cl2O3
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0386609
|
1,8-dichloro-10-[(4-hydroxy-3,5-dimethoxyphenyl)methylidene]anthracen-9-one
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|
C23H16Cl2O4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0415536
|
1,8-dichloro-10-[(3-hydroxy-2,4-dimethoxyphenyl)methylidene]anthracen-9-one
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|
C23H16Cl2O4
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0466409
|
1,8-dichloro-10-[(2-hydroxy-3-methoxyphenyl)methylidene]anthracen-9-one
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|
C22H14Cl2O3
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0386610
|
10-[(2-hydroxy-4-methoxyphenyl)methylidene]anthracen-9-one
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|
C22H16O3
|
1
|
| 1 |
IC50 < 10000 nM
|
|
|
|
CP0415495
|
10-[(3-hydroxyphenyl)methylidene]anthracen-9-one
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|
C21H14O2
|
1
|
| 1 |
IC50 < 10000 nM
|
|
|
