| Compound ID |
Compound Name |
Compound Formula |
|
CP0561124
|
US9062048, 1
Show/Hide
|
C25H27F3N6O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0506926
|
US9062048, 2
Show/Hide
|
C25H30F3N5O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0574870
|
US9062048, 66
Show/Hide
|
C25H27F3N6O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0575633
|
US9062048, 65
Show/Hide
|
C25H27F3N6O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0450158
|
US9062048, 67
Show/Hide
|
C25H27F3N6O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0514981
|
US9062048, 68
Show/Hide
|
C26H29F3N6O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0536317
|
US9062048, 69
Show/Hide
|
C26H28F3N5O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0957710
|
US9062048, 88
Show/Hide
|
C26H31F3N6O2S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0929213
|
US9062048, 89
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0464461
|
US9062048, 7
Show/Hide
|
C24H32F3N5O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0481177
|
US9062048, 9
Show/Hide
|
C22H26F3N5O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0506927
|
US9062048, 10
Show/Hide
|
C24H28F3N5O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0555998
|
US9062048, 70
Show/Hide
|
C25H28F3N7O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0575632
|
US9062048, 62
Show/Hide
|
C25H27F3N6O3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0576452
|
US9062048, 147
Show/Hide
|
C23H25F3N6O2S
|
1
|
| 1 |
IC50 = 9.2 nM
|
|
|
|
CP0464463
|
US9062048, 13
Show/Hide
|
C25H31F3N6O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0555994
|
US9062048, 18
Show/Hide
|
C23H30F3N5O2S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0555591
|
US9062048, 75
Show/Hide
|
C26H29F3N6O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0555584
|
US9062048, 11
Show/Hide
|
C25H29F3N6O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0475261
|
US9062048, 90
Show/Hide
|
C24H32F3N5O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0576451
|
US9062048, 106
Show/Hide
|
C23H28F3N5O3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0518179
|
US9062048, 105
Show/Hide
|
C23H30F3N5O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0239619
|
N-[1-(4-hydroxy-4-phenylcyclohexyl)azetidin-3-yl]-2-[[6-(trifluoromethyl)quinazolin-4-yl]amino]acetamide
Show/Hide
|
C26H28F3N5O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0239620
|
N-[1-(4-phenylcyclohexyl)azetidin-3-yl]-2-[[6-(trifluoromethyl)quinazolin-4-yl]amino]acetamide
Show/Hide
|
C26H28F3N5O
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0557301
|
US9062048, 55
Show/Hide
|
C25H27F3N6O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0575627
|
US9062048, 14
Show/Hide
|
C25H32F3N5O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0488800
|
US9062048, 19
Show/Hide
|
C22H27F3N8O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0555592
|
US9062048, 91
Show/Hide
|
C24H30F3N5O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0555999
|
US9062048, 92
Show/Hide
|
C23H28F3N5O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0904640
|
US9062048, 27
Show/Hide
|
C24H26F3N5O2S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0957361
|
US9062048, 71
Show/Hide
|
C25H28F3N7O
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0450159
|
US9062048, 76
Show/Hide
|
C26H29F3N6O3
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0556094
|
US9062048, 108
Show/Hide
|
C22H28F3N5O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0573992
|
US9062048, 99
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0536318
|
US9062048, 93
Show/Hide
|
C23H30F3N5O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0554189
|
US9062048, 12
Show/Hide
|
C24H29F3N6O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0555590
|
US9062048, 72
Show/Hide
|
C27H27F3N6O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0506769
|
US9062048, 80
Show/Hide
|
C26H31F3N6O2S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0550553
|
US9062048, 81
Show/Hide
|
C23H25F3N6O2S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0318895
|
2-[[2-cyano-6-(trifluoromethyl)quinolin-4-yl]amino]-N-[1-[4-hydroxy-4-(1,3-thiazol-5-yl)cyclohexyl]azetidin-3-yl]acetamide
Show/Hide
|
C25H25F3N6O2S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0920566
|
US9062048, 28
Show/Hide
|
C25H30F3N5O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0555593
|
US9062048, 94
Show/Hide
|
C26H34F3N5O2
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0550552
|
US9062048, 79
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0475265
|
US9062048, 24
Show/Hide
|
C25H25F6N5O2S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0521283
|
US9062048, 100
Show/Hide
|
C25H32F3N5O3
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0536319
|
US9062048, 95
Show/Hide
|
C23H26F3N5O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0961359
|
US9062048, 29
Show/Hide
|
C23H30F3N5O2
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0426600
|
US9062048, 169
Show/Hide
|
C25H33F3N4O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0554190
|
US9062048, 16
Show/Hide
|
C23H27F3N6O3
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0556097
|
US9062048, 111
Show/Hide
|
C23H29F3N6O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0563882
|
US9062048, 51
Show/Hide
|
C24H31F3N6O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0556093
|
US9062048, 63
Show/Hide
|
C32H32F3N5O4S
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0967740
|
US9062048, 87
Show/Hide
|
C24H24F6N6O2S
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0310758
|
N-[1-[4-hydroxy-4-(1,3-thiazol-5-yl)cyclohexyl]azetidin-3-yl]-2-[[6-(trifluoromethyl)quinazolin-4-yl]amino]acetamide
Show/Hide
|
C23H25F3N6O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0555589
|
US9062048, 60
Show/Hide
|
C27H27F3N6O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0578107
|
US9062048, 136
Show/Hide
|
C23H31F3N6O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0563269
|
US9062048, 15
Show/Hide
|
C24H30F3N5O2
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0156848
|
2-[[2,6-bis(trifluoromethyl)quinolin-4-yl]amino]-N-[1-[4-hydroxy-4-(1,3-thiazol-5-yl)cyclohexyl]azetidin-3-yl]acetamide
Show/Hide
|
C25H25F6N5O2S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0957646
|
US9062048, 73
Show/Hide
|
C27H30F3N5O2
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0573848
|
US9062048, 77
Show/Hide
|
C26H29F3N6O3
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0555585
|
US9062048, 20
Show/Hide
|
C23H30F3N5O3
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0556095
|
US9062048, 109
Show/Hide
|
C21H26F3N5O2
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0575629
|
US9062048, 17
Show/Hide
|
C24H29F3N6O3
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0464454
|
US9062048, 101
Show/Hide
|
C20H24F3N5O
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0575630
|
US9062048, 22
Show/Hide
|
C23H27F3N6O3
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0576461
|
US9062048, 52
Show/Hide
|
C24H31F3N6O2
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0563884
|
US9062048, 110
Show/Hide
|
C20H24F3N5O2
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0493321
|
US9062048, 170
Show/Hide
|
C25H31F5N4O2
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0931212
|
US9062048, 134
Show/Hide
|
C24H31F3N6O3S
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0958004
|
US9062048, 26
Show/Hide
|
C24H26F3N5O2S
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0554139
|
US9062048, 34
Show/Hide
|
C22H25F6N5O2
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0524428
|
US9062048, 96
Show/Hide
|
C24H30F3N5O2
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0555995
|
US9062048, 36
Show/Hide
|
C23H28F3N5O
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0554141
|
US9062048, 40
Show/Hide
|
C24H29F3N6O2
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0556098
|
US9062048, 112
Show/Hide
|
C23H26F6N6O2
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0521284
|
US9062048, 119
Show/Hide
|
C21H26F3N5O
|
1
|
| 1 |
IC50 = 82 nM
|
|
|
|
CP0550554
|
US9062048, 120
Show/Hide
|
C24H32F3N5O2
|
1
|
| 1 |
IC50 = 83 nM
|
|
|
|
CP0947431
|
US9062048, 118
Show/Hide
|
C24H33F2N5O
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
|
CP0488804
|
US9062048, 97
Show/Hide
|
C22H28F3N5O2
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0488802
|
US9062048, 58
Show/Hide
|
C26H28F3N5O2
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0561132
|
US9062048, 126
Show/Hide
|
C23H29F3N6O3
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0550555
|
US9062048, 121
Show/Hide
|
C23H30F3N5O2
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0555586
|
US9062048, 25
Show/Hide
|
C25H30F6N4O2
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0488805
|
US9062048, 117
Show/Hide
|
C23H30F3N5O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0488871
|
US9062048, 113
Show/Hide
|
C26H35F3N6O3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0554213
|
US9062048, 122
Show/Hide
|
C24H30F3N5O3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0493303
|
US9062048, 74
Show/Hide
|
C26H30F3N7O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0536030
|
US9062048, 123
Show/Hide
|
C21H23F6N5O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0563883
|
US9062048, 59
Show/Hide
|
C27H27F6N5O2
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0450157
|
US9062048, 33
Show/Hide
|
C25H32F3N5O
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0464466
|
US9062048, 47
Show/Hide
|
C30H35F3N6O3
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0493301
|
US9062048, 38
Show/Hide
|
C25H32F3N5O2
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0554191
|
US9062048, 21
Show/Hide
|
C23H30F3N5O3S
|
1
|
| 1 |
IC50 = 172 nM
|
|
|
|
CP0908190
|
US9062048, 132
Show/Hide
|
C24H31F3N6O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0493307
|
US9062048, 127
Show/Hide
|
C23H29F3N6O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0956357
|
US9062048, 133
Show/Hide
|
C24H31F3N6OS
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0920567
|
US9062048, 30
Show/Hide
|
C25H34F3N5O2
|
1
|
| 1 |
IC50 = 209 nM
|
|
|
|
CP0506928
|
US9062048, 42
Show/Hide
|
C29H33F3N6O3
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0524429
|
US9062048, 124
Show/Hide
|
C24H31F3N6O3
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0550558
|
US9062048, 125
Show/Hide
|
C25H33F3N6O3
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0554140
|
US9062048, 39
Show/Hide
|
C25H31F3N6O2
|
1
|
| 1 |
IC50 = 231 nM
|
|
|
|
CP0563271
|
US9062048, 37
Show/Hide
|
C23H28F3N5O2
|
1
|
| 1 |
IC50 = 235 nM
|
|
|
|
CP0536029
|
US9062048, 116
Show/Hide
|
C21H27F3N6O
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0493258
|
US9062048, 141
Show/Hide
|
C24H32F3N7O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0493254
|
US9062048, 35
Show/Hide
|
C24H25F10N5O2
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0488801
|
US9062048, 57
Show/Hide
|
C24H27F3N6O3
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0561128
|
US9062048, 114
Show/Hide
|
C25H33F3N6O2
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0557300
|
US9062048, 48
Show/Hide
|
C25H33F3N6O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0563270
|
US9062048, 31
Show/Hide
|
C27H34F3N5O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0872143
|
US9062048, 131
Show/Hide
|
C24H29F5N6O
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0468385
|
US9062048, 115
Show/Hide
|
C26H35F3N6O2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0506930
|
US9062048, 53
Show/Hide
|
C23H29F3N6O2
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0956951
|
US9062048, 128
Show/Hide
|
C23H29F3N6O2
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0464464
|
US9062048, 45
Show/Hide
|
C24H31F3N6O2
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0563885
|
US9062048, 129
Show/Hide
|
C30H35F3N6O4
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0550550
|
US9062048, 43
Show/Hide
|
C21H27F3N6O
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0555997
|
US9062048, 44
Show/Hide
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C23H29F3N6O2
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0424176
|
US9062048, 152
Show/Hide
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C23H30F3N5O2
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0506770
|
US9062048, 103
Show/Hide
|
C20H22F3N5O2
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0557302
|
US9062048, 56
Show/Hide
|
C25H31F3N6O2
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0555587
|
US9062048, 41
Show/Hide
|
C22H27F3N6O2
|
1
|
| 1 |
IC50 = 670 nM
|
|
|
|
CP0575631
|
US9062048, 32
Show/Hide
|
C27H38F3N5O2
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0557299
|
US9062048, 23
Show/Hide
|
C24H33F3N6O2
|
1
|
| 1 |
IC50 = 714 nM
|
|
|
|
CP0550551
|
US9062048, 54
Show/Hide
|
C26H33F3N6O2
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0536321
|
US9062048, 98
Show/Hide
|
C25H34F3N5O2
|
1
|
| 1 |
IC50 = 753 nM
|
|
|
|
CP0464465
|
US9062048, 46
Show/Hide
|
C25H33F3N6O2
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0506929
|
US9062048, 50
Show/Hide
|
C24H31F3N6O2
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0908188
|
US9062048, 64
Show/Hide
|
C24H27F3N6O2S
|
1
|
| 1 |
IC50 = 830 nM
|
|
|
|
CP0464455
|
US9062048, 102
Show/Hide
|
C26H34F3N5O
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0493302
|
US9062048, 49
Show/Hide
|
C22H29F3N6O3S
|
1
|
| 1 |
IC50 = 950 nM
|
|
|
|
CP0908189
|
US9062048, 130
Show/Hide
|
C25H31F3N6O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0561134
|
US9062048, 142
Show/Hide
|
C25H34F3N7O2
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0493257
|
US9062048, 139
Show/Hide
|
C24H33F3N6O3S
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0563886
|
US9062048, 138
Show/Hide
|
C25H33F3N6O2
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0577773
|
US9062048, 135
Show/Hide
|
C25H30F6N6O2
|
1
|
| 1 |
IC50 = 2980 nM
|
|
|
|
CP0464456
|
US9062048, 140
Show/Hide
|
C24H30F6N6O3S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0424174
|
US9062048, 137
Show/Hide
|
C25H35F3N6O
|
1
|
| 1 |
IC50 = 5040 nM
|
|
|
|
CP0578108
|
US9062048, 143
Show/Hide
|
C26H36F3N7O2
|
1
|
| 1 |
IC50 = 13840 nM
|
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|
