Brief Information of the Cell Line and Protein
Cell Line ID: CL000040 , THP-1
Synonyms
THP1
THP 1
THPI
THP-1(ATCC)
THP-1-O
O-THP-1
Tohoku Hospital Pediatrics-1
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0006
Protein ID: PT01308 , Tyrosine-protein kinase BTK
Gene Name BTK
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID Q06187
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000040  Protein ID: PT01308
 
Compound ID Compound Name Compound Formula
CP0561590
US9233111, 38
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C31H32FN5O3
 1
1
IC50 = 20 nM
   TI
   LI
   LO
   TS
CP0689423
US9233111, 3
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C31H33FN6O2S
 1
1
IC50 = 27 nM
   TI
   LI
   LO
   TS
CP0442933
US9233111, 16
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C31H33FN6O4
 1
1
IC50 = 69 nM
   TI
   LI
   LO
   TS
CP0132679
US9233111, 62
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C28H34FN7O3
 1
1
IC50 = 71 nM
   TI
   LI
   LO
   TS
CP0564914
US9233111, 24
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C29H29FN4OS
 1
1
IC50 = 94 nM
   TI
   LI
   LO
   TS