| Compound ID |
Compound Name |
Compound Formula |
|
CP0497104
|
imidazopyridine-urea,42
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|
C23H17F4N5O4
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0497102
|
benzimidazole-urea, 16
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|
C23H18F3N5O4
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0497103
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}-2-(2-methoxyethoxy)acetamide
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|
C26H23F4N5O5
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0463179
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}acetamide
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|
C23H17F4N5O3
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0529633
|
benzoxazole-urea, 41
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|
C23H16F4N4O5
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0495693
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}-2-(4-methylpiperazin-1-yl)acetamide
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|
C28H27F4N7O3
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0514246
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}furan-2-carboxamide
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|
C26H17F4N5O4
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0372460
|
N-(6-{[6-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)pyridin-3-yl]oxy}-1H-1,3-benzodiazol-2-yl)acetamide
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|
C22H16F4N6O3
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
|
CP0503137
|
imidazopyridine-urea, 43
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|
C22H16F4N6O4
|
1
|
| 1 |
IC50 = 6.5 nM
|
|
|
|
CP0514248
|
benzthiazole-urea, 40
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|
C23H16F4N4O4S
|
1
|
| 1 |
IC50 = 7.2 nM
|
|
|
|
CP0372463
|
benzimidazole-urea, 20
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|
C22H18BrN5O4
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0258617
|
benzimidazole-urea, 17
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|
C23H17F4N5O4
|
1
|
| 1 |
IC50 = 8.7 nM
|
|
|
|
CP0464614
|
benzimidazole-urea, 18
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|
C23H17ClF3N5O4
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0463178
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}pyridine-3-carboxamide
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|
C27H18F4N6O3
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0372458
|
benzimidazole-urea, 38
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|
C24H19F4N5O4
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0372462
|
benzimidazole-urea, 23
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|
C23H18F3N5O4S
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0532174
|
benzimidazole-urea, 21
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|
C22H18ClN5O4
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0514251
|
benzimidazole-urea, 24
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|
C23H21N5O4S
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0532173
|
benzimidazole-urea, 35
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|
C23H17F4N5O4S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0503138
|
benzimidazole-urea, 22
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|
C22H17F2N5O4
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0497105
|
benzimidazole-urea, 34
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|
C23H17F4N5O3S
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0497106
|
benzimidazole-urea, 30
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|
C23H17F4N5O4
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0514250
|
benzimidazole-urea, 31
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|
C22H16F4N6O4
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0495714
|
imidazopyridine-urea, 44
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|
C22H16F4N6O4
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0529632
|
N-{6-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1H-1,3-benzodiazol-2-yl}benzamide
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|
C28H19F4N5O3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0372459
|
benzimidazole-urea, 36
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|
C23H17F4N5O5S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0020880
|
benzimidazole-urea, 19
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|
C24H23N5O4
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0514249
|
5-({[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl}amino)-2-({2-[(methoxycarbonyl)amino]-1H-1,3-benzodiazol-6-yl}oxy)-1-oxidopyridin-1-ium
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|
C22H16F4N6O5
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0372457
|
3-[2-fluoro-5-(trifluoromethyl)phenyl]-1-{4-[(2-{[2-(4-methylpiperazin-1-yl)ethyl]amino}-1H-1,3-benzodiazol-6-yl)oxy]phenyl}urea
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|
C28H29F4N7O2
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0497107
|
benzimidazole-thiourea, 27
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|
C23H18F3N5O3S
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0514247
|
1-{4-[(2-amino-1H-1,3-benzodiazol-6-yl)oxy]phenyl}-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea
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|
C21H15F4N5O2
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
