Brief Information of the Cell Line and Protein
Cell Line ID: CL000027 , tsA201
Synonyms
tsA-201
HEK293-TSA
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_2737
Protein ID: PT02031 , Voltage-dependent N-type calcium channel subunit alpha-1B
Gene Name CACNA1B
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID Q00975
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000027  Protein ID: PT02031
 
Compound ID Compound Name Compound Formula
CP0024074
(2R)-2-[[6-[(5-methylthiophen-2-yl)methylamino]-9-propylpurin-2-yl]amino]butan-1-ol
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C18H26N6OS
 1
1
EC50 = 7210 nM
   TI
   LI
   LO
   TS
CP0025048
(2R)-2-[[6-[(5-methylthiophen-2-yl)methylamino]-9-propan-2-ylpurin-2-yl]amino]butan-1-ol
   Show/Hide
C18H26N6OS
 1
1
EC50 = 11290 nM
   TI
   LI
   LO
   TS
CP0022076
(2R)-2-[[6-(benzylamino)-9-propylpurin-2-yl]amino]butan-1-ol
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C19H26N6O
 1
1
EC50 = 14230 nM
   TI
   LI
   LO
   TS
CP0001111
(2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]amino]butan-1-ol
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C19H26N6O
 1
1
EC50 = 27580 nM
   TI
   LI
   LO
   TS
CP0024075
(2R)-2-[[9-methyl-6-[(5-methylthiophen-2-yl)methylamino]purin-2-yl]amino]butan-1-ol
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C16H22N6OS
 1
1
EC50 = 30020 nM
   TI
   LI
   LO
   TS
CP0016234
(2R)-2-[[6-(benzylamino)-9-methylpurin-2-yl]amino]butan-1-ol
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C17H22N6O
 1
1
EC50 > 70000 nM
   TI
   LI
   LO
   TS
CP0008732
OLOMOUCINE II
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C19H26N6O2
 1
1
EC50 = 80000 nM
   TI
   LI
   LO
   TS
CP0016230
(2R)-2-[[6-(benzhydrylamino)-9-propan-2-ylpurin-2-yl]amino]butan-1-ol
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C25H30N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0016231
(2R)-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-ylpurin-2-yl]amino]butan-1-ol
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C25H30N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0016232
(2R)-2-[[9-methyl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]butan-1-ol
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C16H21N7O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0016233
(2R)-2-[[6-[(4-phenylphenyl)methylamino]-9-propylpurin-2-yl]amino]butan-1-ol
   Show/Hide
C25H30N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0017275
(2R)-2-[[9-propyl-6-[[4-(trifluoromethyl)phenyl]methylamino]purin-2-yl]amino]butan-1-ol
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C20H25F3N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0017346
(2R)-2-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]butan-1-ol
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C18H25N7O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0017347
(2R)-2-[[6-(2-phenylethylamino)-9-propylpurin-2-yl]amino]butan-1-ol
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C20H28N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0017348
(2R)-2-[[6-(cyclopropylmethylamino)-9-propylpurin-2-yl]amino]butan-1-ol
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C16H26N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0019896
(2R)-2-[[6-(cyclopropylmethylamino)-9-propan-2-ylpurin-2-yl]amino]butan-1-ol
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C16H26N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0019897
(2R)-2-[[9-propyl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]butan-1-ol
   Show/Hide
C18H25N7O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0022073
(2R)-2-[[6-(cyclopropylmethylamino)-9-methylpurin-2-yl]amino]butan-1-ol
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C14H22N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0022074
(2R)-2-[[9-methyl-6-(2-phenylethylamino)purin-2-yl]amino]butan-1-ol
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C18H24N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0022075
(2R)-2-[[6-(benzhydrylamino)-9-propylpurin-2-yl]amino]butan-1-ol
   Show/Hide
C25H30N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0024076
(2R)-2-[[6-(2-phenylethylamino)-9-propan-2-ylpurin-2-yl]amino]butan-1-ol
   Show/Hide
C20H28N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0025153
(2R)-2-[(6-anilino-9-propylpurin-2-yl)amino]butan-1-ol
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C18H24N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0025480
(2R)-2-[[6-(benzhydrylamino)-9-methylpurin-2-yl]amino]butan-1-ol
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C23H26N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0030457
(2R)-2-[[9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methylamino]purin-2-yl]amino]butan-1-ol
   Show/Hide
C20H25F3N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0030458
(2R)-2-[(6-anilino-9-methylpurin-2-yl)amino]butan-1-ol
   Show/Hide
C16H20N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0030459
(2R)-2-[[9-methyl-6-[(4-phenylphenyl)methylamino]purin-2-yl]amino]butan-1-ol
   Show/Hide
C23H26N6O
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0007240
(2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol
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C19H26N6O
 1
1
EC50 < 100000 nM
   TI
   LI
   LO
   TS